SCHEMBL7084465

SCHEMBL7084465

OC(CCc1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)cn1)c1ccc2ccccc2c1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 13/20 0.44
HDAC1 Q13547 2/20 0.38
HDAC8 Q9BY41 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
HTR1A P08908 1/20 0.37
AOC3 Q16853 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
TSHR P16473 1/20 0.37
HIF1A Q16665 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8979144 0.84 SIRT2 (0.42) SIRT2HTR1A
SCHEMBL4033379 0.81 HDAC1 (0.43) SIRT2HDAC1
SCHEMBL9258121 0.76 SIRT2 (0.42) SIRT2
SCHEMBL6964092 0.75 SIRT2 (0.38) SIRT2
SCHEMBL7080830 0.75 SIRT2 (0.44) SIRT2HDAC1HDAC8
SCHEMBL4025341 0.74 SIRT2 (0.47) SIRT2
SCHEMBL1037984 0.73 SIRT2 (0.40) SIRT2
SCHEMBL6958792 0.73 SIRT2 (0.38) SIRT2
SCHEMBL1041048 0.73 SIRT2 (0.49) SIRT2
SCHEMBL19865793 0.71 SIRT2 (0.50) SIRT2MEN1KMT2ACYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0974584-B1 FUSED RING COMPOUNDS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-01-15 EP disclosed
US-6420375-B1 ANTITUMOR TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-16 US disclosed
EP-0974584-A1 FUSED RING COMPOUNDS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-01-26 EP disclosed