SCHEMBL7085115

SCHEMBL7085115

CC(C)c1nc(CCOC(N)=O)n(Cc2ccncc2)c1Sc1cccc(F)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 4/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
PIM1 P11309 2/20 0.33
PIM3 Q86V86 1/20 0.33
CYP3A4 P08684 3/20 0.32
CYP2D6 P10635 3/20 0.32
CYP2C9 P11712 3/20 0.32
CYP1A2 P05177 2/20 0.32
CYP2C19 P33261 2/20 0.32
EPHX1 P07099 1/20 0.31
USP2 O75604 2/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
MAPT P10636 1/20 0.31
CDC7 O00311 1/20 0.31
ROCK2 O75116 1/20 0.31
MAP4K4 O95819 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972238 0.95 PPARG (0.34) ENPP2GRIN1GRIN2BLMNATP53
SCHEMBL7082343 0.93 GRIN1 (0.32) ENPP2GRIN1GRIN2BLMNATP53
SCHEMBL6975545 0.92 GRIN1 (0.34) ENPP2GRIN1GRIN2BLMNATP53
SCHEMBL6967988 0.92 ENPP2 (0.35) ENPP2TP53PIM1PIM3
SCHEMBL6973183 0.91 ENPP2 (0.35) ENPP2GRIN1GRIN2BLMNATP53
SCHEMBL7080841 0.91 GRIN1 (0.36) ENPP2GRIN1GRIN2BLMNAALDH1A1
SCHEMBL6961900 0.91 PIM1 (0.35) LMNATP53PIM1PIM3ALDH1A1
SCHEMBL6968774 0.89 PIM1 (0.35) ENPP2LMNAPIM1PIM3CYP3A4
SCHEMBL6973633 0.88 EPHX1 (0.34) LMNAEPHX1ALDH1A1MAPTSLC6A9
SCHEMBL6965758 0.87 ENPP2 (0.34) ENPP2LMNAPIM1PIM3GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed