SCHEMBL6975545

SCHEMBL6975545

CC(=O)OCCc1nc(C(C)C)c(Sc2cccc(F)c2)n1Cc1ccncc1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
ENPP2 Q13822 4/20 0.34
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
CYP3A4 P08684 3/20 0.32
CYP2D6 P10635 3/20 0.32
CYP2C9 P11712 3/20 0.32
CYP1A2 P05177 2/20 0.32
CYP2C19 P33261 2/20 0.32
USP2 O75604 2/20 0.32
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
MAPT P10636 1/20 0.31
SLC6A9 P48067 2/20 0.31
CYP19A1 P11511 1/20 0.31
PPARG P37231 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7086007 0.93 GRIN1 (0.33) GRIN1GRIN2BENPP2LMNATP53
SCHEMBL7085115 0.92 ENPP2 (0.33) GRIN1GRIN2BENPP2LMNATP53
SCHEMBL6969213 0.92 ENPP2 (0.35) ENPP2TP53CYP19A1PPARG
SCHEMBL6973952 0.91 ENPP2 (0.36) GRIN1GRIN2BENPP2LMNATP53
SCHEMBL6960486 0.90 IDO1 (0.34) LMNATP53MAPTSLC6A9
SCHEMBL6972238 0.87 PPARG (0.34) GRIN1GRIN2BENPP2LMNATP53
SCHEMBL6974529 0.87 DHODH (0.34) LMNACYP2C9CYP1A2CYP2C19ALDH1A1
SCHEMBL8347170 0.87 TBXA2R (0.42) GRIN1GRIN2BENPP2LMNATP53
SCHEMBL7086066 0.87 KMT2A (0.36) LMNACYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL6974113 0.86 S1PR3 (0.38) GRIN1GRIN2BSLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed