SCHEMBL6965758

SCHEMBL6965758

CC(C)c1nc(CCCOC(N)=O)n(Cc2ccncc2)c1Sc1cc(F)cc(F)c1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 3/20 0.34
PPARG P37231 6/20 0.33
GSK3B P49841 1/20 0.32
AGTR1 P30556 2/20 0.32
AGTR2 P50052 2/20 0.32
LMNA P02545 1/20 0.31
PIM1 P11309 1/20 0.31
PIM3 Q86V86 1/20 0.31
TLR7 Q9NYK1 2/20 0.31
KCNH2 Q12809 1/20 0.31
CYP19A1 P11511 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967988 0.95 ENPP2 (0.35) ENPP2PIM1PIM3CYP19A1MEN1
SCHEMBL6972238 0.93 PPARG (0.34) ENPP2PPARGGSK3BAGTR1AGTR2
SCHEMBL6972000 0.92 MEN1 (0.33) GSK3BLMNACYP19A1MEN1KMT2A
SCHEMBL6971875 0.92 LMNA (0.41) PPARGGSK3BAGTR1AGTR2LMNA
SCHEMBL6973533 0.92 LMNA (0.34) GSK3BLMNACYP19A1
SCHEMBL6961399 0.91 PPARG (0.35) ENPP2PPARGAGTR1AGTR2LMNA
SCHEMBL6961792 0.91 ENPP2 (0.32) ENPP2PIM1PIM3CYP19A1
SCHEMBL6968648 0.90 P2RX3 (0.33) PPARGGSK3BLMNAPIM1PIM3
SCHEMBL6971680 0.90 PIM1 (0.33) ENPP2PPARGGSK3BLMNAPIM1
SCHEMBL6970826 0.90 GRIN1 (0.35) ENPP2LMNATLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed