SCHEMBL708527

SCHEMBL708527

O=C(O)c1cc2c(Cl)c(Cl)ccc2[nH]1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 4/20 0.57
HRH4 Q9H3N8 1/20 0.57
KDM4E B2RXH2 3/20 0.54
LMNA P02545 2/20 0.54
ALDH1A1 P00352 2/20 0.54
HSD17B10 Q99714 2/20 0.54
RHEB Q15382 4/20 0.54
F7 P08709 1/20 0.53
F3 P13726 1/20 0.53
EIF4A3 P38919 1/20 0.50
MEN1 O00255 3/20 0.49
HPGD P15428 3/20 0.49
KMT2A Q03164 3/20 0.49
MAPK1 P28482 2/20 0.49
CYP2C9 P11712 2/20 0.49
BLM P54132 2/20 0.49
NGFR P08138 1/20 0.49
GRIN2D O15399 3/20 0.49
GRIN3B O60391 3/20 0.49
GRIN2A Q12879 3/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29425136 0.83 DAO (0.58) GRIN1KDM4ELMNAALDH1A1HSD17B10
SCHEMBL11740631 0.83 KDM4E (0.51) GRIN1HRH4KDM4ELMNAALDH1A1
SCHEMBL1504212 0.83 HRH4 (0.59) GRIN1HRH4KDM4ELMNAALDH1A1
SCHEMBL6161388 0.83 DAO (0.58) GRIN1KDM4ELMNAALDH1A1HSD17B10
SCHEMBL3096730 0.83 GRIN1 (0.54) GRIN1HRH4KDM4ELMNAALDH1A1
SCHEMBL6168680 0.82 MEN1 (0.58) HRH4KDM4ELMNAALDH1A1HSD17B10
SCHEMBL24754486 0.80 HRH4 (0.56) HRH4RHEBKMT2AALOX15
SCHEMBL19331400 0.80 HRH4 (0.56) HRH4KDM4EALDH1A1HSD17B10HPGD
SCHEMBL30039640 0.80 HRH4 (0.56) HRH4KDM4EALDH1A1HSD17B10HPGD
SCHEMBL3110626 0.79 KDM4E (0.59) GRIN1KDM4ELMNAALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 39 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4747234-A1 KV1.3 POTASSIUM CHANNEL ANTAGONISTS Muna Therapeutics ApS (DK) 2026-05-27 EP disclosed
EP-4747235-A1 KV1.3 POTASSIUM CHANNEL ANTAGONISTS Muna Therapeutics ApS (DK) 2026-05-27 EP disclosed
EP-3976617-B1 FUSED HETEROCYCLIC DERIVATIVES JANSSEN SCIENCES IRELAND UNLIMITED CO (IE) 2025-04-23 EP disclosed
WO-2025017103-A1 KV1.3 POTASSIUM CHANNEL ANTAGONISTS MUNA THERAPEUTICS APS (DK) 2025-01-23 WO disclosed
WO-2025017105-A1 KV1.3 POTASSIUM CHANNEL ANTAGONISTS MUNA THERAPEUTICS APS (DK) 2025-01-23 WO disclosed
US-20220348592-A1 FUSED HETEROCYCLIC DERIVATIVES JANSSEN PHARMACEUTICA NV (BE) 2022-11-03 US disclosed
EP-3976617-A1 FUSED HETEROCYCLIC DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2022-04-06 EP disclosed
CN-113906028-A Fused heterocyclic derivatives 爱尔兰詹森科学公司 2022-01-07 CN disclosed
WO-2020243135-A1 FUSED HETEROCYCLIC DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2020-12-03 WO disclosed
WO-2020243135-A1 FUSED HETEROCYCLIC DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2020-12-03 WO disclosed
US-20040132715-A1 Method to treat allergic rhinitis DUNFORD PAUL J (US) 2004-07-08 US disclosed
WO-2004022061-A1 USE OF INDOLYL DERIVATIVES FOR THE MANUFACTURE OF A MEDICAMENT FOR THE TREATMENT ALLERGIC RHINITIS JANSSEN PHARMACEUTICA, N.V. (BE) 2004-03-18 WO disclosed
EP-1373204-A2 HETEROCYCLIC COMPOUNDS Ortho-McNeil Pharmaceutical, Inc. (US) 2004-01-02 EP disclosed
US-20030207893-A1 Heterocyclic compounds ORTHO MCNEIL PHARMACEUTICAL, INC. 2003-11-06 US disclosed
US-6608070-B1 Useful for treatment of medical condition in which prostaglandins are implicated as pathogens NAKAO KAZUNARI (JP) 2003-08-19 US disclosed
WO-2002072548-A2 HETEROCYCLIC COMPOUNDS AND THEIR USE AS HISTAMINE H4 LIGANDS. ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2002-09-19 WO disclosed
EP-1045833-A1 2,3-SUBSTITUTED INDOLE COMPOUNDS AS COX-2 INHIBITORS PFIZER INC. (US) 2000-10-25 EP disclosed
CN-1265591-A Coumpound ZENECA LTD (GB) 2000-09-06 CN disclosed
WO-1999035130-A1 2,3-SUBSTITUTED INDOLE COMPOUNDS AS COX-2 INHIBITORS PFIZER PHARMACEUTICALS INC. (JP) 1999-07-15 WO disclosed
US-4060626-A Indole-carboxylic carbon compounds and pharmaceutical compositions containing them BOEHRINGER MANNHEIM G.M.B.H. (DT) 1977-11-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220348592-A1 FUSED HETEROCYCLIC DERIVATIVES HAVCR2, HCCS, GOT2 GRIN1 3749/4885HRH4 888/4885KDM4E 3515/4885
US-20040132715-A1 Method to treat allergic rhinitis HRH2, HRH4, HRH1 GRIN1 1051/4885HRH4 2/4885KDM4E 3580/4885
US-20030207893-A1 Heterocyclic compounds AADAC, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, NQO1 GRIN1 2264/4885HRH4 1508/4885KDM4E 3201/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.