SCHEMBL7085528

SCHEMBL7085528

C#CCC(=O)c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.58
TDP1 Q9NUW8 3/20 0.58
MAPT P10636 3/20 0.58
KMT2A Q03164 3/20 0.58
CES1 P23141 3/20 0.58
MEN1 O00255 2/20 0.58
CYP3A4 P08684 2/20 0.58
HPGD P15428 2/20 0.58
KDM4E B2RXH2 1/20 0.58
ALOX15 P16050 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
ALDH1A1 P00352 6/20 0.54
GSK3B P49841 2/20 0.54
PTPN1 P18031 2/20 0.54
HIF1A Q16665 2/20 0.54
TRPA1 O75762 1/20 0.54
L3MBTL1 Q9Y468 2/20 0.52
LMNA P02545 2/20 0.52
NR4A2 P43354 1/20 0.52
ERCC5 P28715 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzene SCHEMBL28690163 1.00 MAPK1 (0.58) MAPK1TDP1MAPTKMT2ACES1
SCHEMBL8657431 0.94 MAPT (0.52) MAPK1TDP1MAPTKMT2ACES1
Fluorobenzene SCHEMBL28684421 0.90 HSD11B1 (0.49) MAPK1TDP1MAPTKMT2ACES1
Anisole SCHEMBL28690179 0.85 L3MBTL1 (0.54) TDP1MAPTKMT2ACES1MEN1
SCHEMBL3629497 0.81 ALDH1A1 (0.63) MAPK1TDP1MAPTKMT2ACES1
SCHEMBL29087821 0.81 POLB (0.49) MAPK1TDP1MAPTKMT2ACES1
SCHEMBL571114 0.81 TDP1 (0.58) MAPK1TDP1MAPTKMT2ACES1
SCHEMBL10556922 0.80 TDP1 (0.57) MAPK1TDP1MAPTKMT2ACES1
SCHEMBL22313390 0.79 CES1 (0.56) MAPK1TDP1MAPTKMT2ACES1
SCHEMBL136826 0.79 CES1 (0.56) MAPK1TDP1MAPTKMT2ACES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1294699-B1 MODULATORS OF TNF- ALPHA SIGNALLING GENZYME CORP (US) 2016-04-13 EP claimed
EP-1051413-B1 QUINOLINE DERIVATIVES AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2003-06-04 EP claimed
EP-0548664-B1 2,3,3a-5,9b-hexahydro-1H-benzo(e)indole derivatives HOFFMANN LA ROCHE (CH) 1995-05-31 EP claimed
CN-114057623-B N-naphthyl indole derivative and synthesis method thereof 湖南第一师范学院 2023-07-21 CN disclosed
CN-114057623-A N-naphthyl indole derivative and synthetic method thereof 湖南第一师范学院 2022-02-18 CN disclosed
WO-2008018063-A2 TETRAARYLPORPHINE DERIVATIVES AND USES THEREOF KODESH S.A (LU) 2008-02-14 WO disclosed