SCHEMBL7085698

SCHEMBL7085698

Nc1ccc(N)c(-c2ccnc(C(F)(F)F)c2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.44
IDO1 P14902 1/20 0.44
MAP4K4 O95819 1/20 0.44
LOXL2 Q9Y4K0 2/20 0.44
LOX P28300 1/20 0.42
PARP15 Q460N3 1/20 0.41
PARP14 Q460N5 1/20 0.41
PARP10 Q53GL7 1/20 0.41
TIPARP Q7Z3E1 1/20 0.41
PARP16 Q8N5Y8 1/20 0.41
PARP11 Q9NR21 1/20 0.41
GLA P06280 1/20 0.38
POLB P06746 1/20 0.38
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.38
SYK P43405 2/20 0.37
CA2 P00918 1/20 0.37
CHKA P35790 1/20 0.37
LRRK2 Q5S007 1/20 0.36
ALOX5AP P20292 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27195309 0.86 NOS3 (0.46) NOTUMIDO1MAP4K4LOXL2LOX
SCHEMBL7088779 0.78 ADORA2B (0.49) IDO1MAP4K4LOXL2PARP10PARP11
SCHEMBL23910018 0.78 CYP3A4 (0.47) NOTUMIDO1MAP4K4LOXL2LOX
SCHEMBL7088884 0.78 DYRK1A (0.43) NOS3NOS2DYRK1A
SCHEMBL7085072 0.77 KCNH2 (0.50) MAP4K4GLAPOLBGAATSHR
SCHEMBL29418957 0.77 LOXL2 (0.57) NOTUMIDO1MAP4K4LOXL2LOX
SCHEMBL111794 0.77 LOXL2 (0.57) NOTUMIDO1MAP4K4LOXL2LOX
SCHEMBL23916460 0.76 PARP15 (0.39) NOTUMIDO1MAP4K4LOXL2LOX
SCHEMBL7085158 0.75 KDM4C (0.42) MAP4K4POLBGAAAAK1
SCHEMBL7086532 0.75 CCNC (0.43) MAP4K4DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1052252-B1 Diaminobenzene derivatives and dyeing preparations containing them WELLA AG (DE) 2003-08-06 EP claimed
US-6461388-B1 Diaminobenzene derivative compounds and dye compositions containing same WELLA AKTIENGESELLSCHAFT (DE) 2002-10-08 US claimed
EP-1052252-A1 Diaminobenzene derivatives and dyeing preparations containing them Wella Aktiengesellschaft (DE) 2000-11-15 EP claimed
EP-1052252-B1 Diaminobenzene derivatives and dyeing preparations containing them WELLA AG (DE) 2003-08-06 EP disclosed
US-6461388-B1 Diaminobenzene derivative compounds and dye compositions containing same WELLA AKTIENGESELLSCHAFT (DE) 2002-10-08 US disclosed
EP-1052252-A1 Diaminobenzene derivatives and dyeing preparations containing them Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed