SCHEMBL7086513

SCHEMBL7086513

CC(C)c1nc(CNS(C)(=O)=O)n(Cc2ccccn2)c1Sc1cccc(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
POLB P06746 3/20 0.36
LMNA P02545 1/20 0.35
HPGD P15428 1/20 0.34
GRM5 P41594 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TP53 P04637 1/20 0.34
ALDH1A1 P00352 3/20 0.33
GRM4 Q14833 1/20 0.33
AGTR1 P30556 1/20 0.33
THRB P10828 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
MAPT P10636 1/20 0.33
PPP1CA P62136 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973271 0.93 POLB (0.35) POLBHPGDSMN1; SMN2TP53ALDH1A1
SCHEMBL8508399 0.92 LMNA (0.36) GRIN1GRIN2BPOLBLMNAGRM5
SCHEMBL7077261 0.90 POLB (0.35) POLBLMNAALDH1A1THRBKMT2A
SCHEMBL6974276 0.90 GRIN1 (0.37) GRIN1GRIN2BALDH1A1GRM4ADORA2A
SCHEMBL6961462 0.88 GRIN1 (0.37) GRIN1GRIN2BPOLBHPGDGRM5
SCHEMBL6969739 0.87 POLB (0.38) GRIN1GRIN2BPOLBHPGDTP53
SCHEMBL6972096 0.87 LMNA (0.37) POLBLMNASMN1; SMN2TP53ALDH1A1
SCHEMBL6974408 0.87 L3MBTL1 (0.44) POLBLMNASMN1; SMN2TP53ALDH1A1
SCHEMBL7085418 0.86 POLB (0.38) GRIN1GRIN2BPOLBHPGDTP53
SCHEMBL7080069 0.86 S1PR3 (0.37) GRIN1GRIN2BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed