SCHEMBL7086916

SCHEMBL7086916

NC(=O)C=Cc1ccc2nc(Nc3ccccc3)ncc2n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C9 P11712 2/20 0.43
MEN1 O00255 1/20 0.43
USP2 O75604 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
CYP2C19 P33261 1/20 0.43
KMT2A Q03164 1/20 0.43
SYK P43405 1/20 0.43
AURKA O14965 3/20 0.43
JAK2 O60674 1/20 0.43
AURKB Q96GD4 1/20 0.43
GSK3B P49841 4/20 0.41
GSK3A P49840 3/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
BRAF P15056 1/20 0.41
EGFR P00533 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7086914 1.00 CYP1A2 (0.43) CYP1A2CYP3A4CYP2C9MEN1USP2
SCHEMBL1262019 0.75 MKNK2 (0.53) MAPK1AURKBKDM4EBRAFEGFR
SCHEMBL1262018 0.75 MKNK2 (0.53) MAPK1AURKBKDM4EBRAFEGFR
SCHEMBL7086918 0.74 SYK (0.46) CYP1A2CYP3A4CYP2C9MEN1USP2
SCHEMBL30209645 0.71 KDM4E (0.56) CYP1A2CYP2C9MEN1CYP2C19KMT2A
SCHEMBL4716351 0.70 GSK3B (0.47) MEN1TSHRMAPK1KMT2ASYK
SCHEMBL4716354 0.70 GSK3B (0.47) MEN1TSHRMAPK1KMT2ASYK
SCHEMBL12120895 0.70 JAK2 (0.51) CYP1A2CYP3A4CYP2C9MEN1USP2
SCHEMBL7060640 0.70 ABCG2 (0.54) MAPK1AURKBEGFRMAP4K4PIM1
SCHEMBL5717630 0.70 LMNA (0.73) CYP1A2MEN1MAPK1CYP2C19KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1366027-A1 COMBI-MOLECULES HAVING SIGNAL TRANSDUCTION INHIBITORY PROPERTIES AND DNA DAMAGING PROPERTIES McGILL UNIVERSITY (CA) 2003-12-03 EP disclosed
WO-2002068396-A1 COMBI-MOLECULES HAVING SIGNAL TRANSDUCTION INHIBITORY PROPERTIES AND DNA DAMAGING PROPERTIES MCGILL UNIVERSITY (CA) 2002-09-06 WO disclosed