SCHEMBL7087593

SCHEMBL7087593

Cc1cc(C(C)Br)n(O)c(=O)c1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 17/20 0.44
NR1I2 O75469 1/20 0.41
KDM4B O94953 1/20 0.41
CHRM1 P11229 1/20 0.41
TBXA2R P21731 1/20 0.41
ADRA1A P35348 1/20 0.41
DOHH Q9BU89 1/20 0.41
DAO P14920 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7087619 0.84 IDH1 (0.46) IDH1NR1I2KDM4BCHRM1TBXA2R
SCHEMBL11852460 0.75 IDH1 (0.54) IDH1
SCHEMBL10730246 0.73 IDH1 (0.51) IDH1NR1I2KDM4BCHRM1TBXA2R
SCHEMBL11848025 0.72 NR1I2 (0.55) IDH1NR1I2KDM4BCHRM1TBXA2R
SCHEMBL21762069 0.70 IDH1 (0.42) IDH1NR1I2KDM4BCHRM1TBXA2R
SCHEMBL10726848 0.70 IDH1 (0.42) IDH1NR1I2KDM4BCHRM1TBXA2R
SCHEMBL11435622 0.70 IDH1 (0.49) IDH1NR1I2KDM4BCHRM1TBXA2R
Metipirox SCHEMBL794955 0.70 IDH1 (0.52) IDH1NR1I2KDM4BCHRM1TBXA2R
SCHEMBL10729237 0.68 IDH1 (0.40) IDH1NR1I2KDM4BCHRM1TBXA2R
SCHEMBL10724185 0.68 IDH1 (0.47) IDH1NR1I2KDM4BCHRM1TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030228340-A1 Methods for treating rosacea with pyridones MEDICIS PHARMACEUTICAL CORPORATION 2003-12-11 US disclosed
WO-2003084538-A1 METHODS FOR TREATING ROSACEA WITH PYRIDONES MEDICIS PHARMACEUTICAL CORPORATION (US) 2003-10-16 WO disclosed