SCHEMBL7089113

SCHEMBL7089113

Cc1ccc(N)cc1CCN1CCC(c2c[nH]c3c(Cl)cccc23)CC1.Cc1ccc(N)cc1CCN1CCC(c2c[nH]c3cc(Cl)ccc23)CC1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.47
OPRK1 P41145 3/20 0.47
OPRL1 P41146 3/20 0.47
HTR6 P50406 2/20 0.45
KCNH2 Q12809 2/20 0.45
SLC6A4 P31645 2/20 0.42
DRD2 P14416 1/20 0.42
HTR1D P28221 1/20 0.41
HTR1B P28222 1/20 0.41
CCR2 P41597 1/20 0.40
ADRA1D P25100 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6593968 0.92 OPRM1 (0.54) OPRM1OPRK1OPRL1HTR6KCNH2
SCHEMBL6598131 0.91 SLC6A4 (0.49) OPRM1OPRK1OPRL1HTR6KCNH2
SCHEMBL6596780 0.84 HTR1D (0.56) OPRM1OPRK1OPRL1HTR6KCNH2
SCHEMBL27537908 0.78 OPRM1 (0.50) OPRM1OPRK1OPRL1HTR6KCNH2
SCHEMBL27541443 0.77 APP (0.50) OPRM1OPRK1OPRL1HTR6KCNH2
SCHEMBL6598134 0.77 HTR1D (0.50) OPRM1OPRK1OPRL1DRD2HTR1D
SCHEMBL31143224 0.77 ADRA1D (0.57) OPRM1OPRK1OPRL1HTR6KCNH2
SCHEMBL6598294 0.76 HTR1D (0.45) SLC6A4DRD2HTR1DHTR1BCCR2
SCHEMBL6595114 0.76 OPRM1 (0.48) OPRM1OPRK1OPRL1DRD2HTR1D
SCHEMBL6598237 0.76 OPRM1 (0.47) OPRM1OPRK1OPRL1SLC6A4HTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1305307-A1 INDOLE DERIVATIVES USEFUL FOR THE TREATMENT OF CNS DISORDERS H. Lundbeck A/S (DK) 2003-05-02 EP disclosed
WO-2002008223-A1 INDOLE DERIVATIVES USEFUL FOR THE TREATMENT OF CNS DISORDERS H. LUNDBECK A/S (DK) 2002-01-31 WO disclosed