SCHEMBL7090107

SCHEMBL7090107

Cc1ccc(Nc2n[nH]c(Sc3ccc(Br)s3)n2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.42
RAB9A P51151 5/20 0.42
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
MAPT P10636 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
TSHR P16473 1/20 0.42
NFKB1 P19838 1/20 0.42
CASP3 P42574 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
LMNA P02545 1/20 0.39
GAA P10253 3/20 0.35
MAPK1 P28482 1/20 0.35
METAP2 P50579 3/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7085921 0.87 CDC7 (0.38) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL7083924 0.87 MAPT (0.44) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL7089497 0.85 PIK3CA (0.42) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL7084630 0.85 MEN1 (0.42) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL5385647 0.81 METAP2 (0.42) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL7080965 0.80 SMN1; SMN2 (0.41) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL7087741 0.77 CDK2 (0.43) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL7084060 0.75 ALDH1A1 (0.44) NPC1RAB9AKMT2AMAPTSMN1; SMN2
SCHEMBL7087201 0.74 RAB9A (0.42) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL7084268 0.73 MAPT (0.46) NPC1RAB9AMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1223932-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2003-01-15 EP claimed
EP-1223932-A1 COMPOUNDS AND METHODS SmithKline Beecham Corporation (US) 2002-07-24 EP claimed
WO-2001024796-A1 1,2,4-TRIAZOLE DERIVATIVES, COMPOSITION, PROCESS OF MAKING AND METHODS OF USE SMITHKLINE BEECHAM CORPORATION (US) 2001-04-12 WO claimed