SCHEMBL7090123

SCHEMBL7090123

COc1ccc(N)cc1C1OCCO1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.42
ALDH1A1 P00352 6/20 0.42
USP2 O75604 1/20 0.42
MAPT P10636 4/20 0.41
CYP19A1 P11511 3/20 0.41
GAA P10253 2/20 0.41
LMNA P02545 1/20 0.41
TSHR P16473 2/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
NR4A1 P22736 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
GFER P55789 1/20 0.39
CYP2C19 P33261 1/20 0.38
NR3C1 P04150 1/20 0.37
DRD4 P21917 1/20 0.37
MEN1 O00255 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL829699 0.86 MAPT (0.44) KDM4EALDH1A1USP2MAPTCYP19A1
SCHEMBL5259483 0.85 MAPT (0.43) KDM4EALDH1A1USP2MAPTCYP19A1
SCHEMBL27664506 0.84 SMN1; SMN2 (0.38) KDM4EALDH1A1USP2MAPTCYP19A1
SCHEMBL7093467 0.81 ACHE (0.48) ALDH1A1USP2MAPTGAALMNA
SCHEMBL1670216 0.79 MEN1 (0.47) KDM4EALDH1A1GAATSHRHTT
SCHEMBL7053663 0.79 NPC1 (0.39) ALDH1A1MAPK1NPC1RAB9ACYP2C19
SCHEMBL7819793 0.79 GRIN2B (0.31) GAATSHR
SCHEMBL7093466 0.77 NPC1 (0.42) ALDH1A1MAPTGAALMNATSHR
SCHEMBL7938441 0.77 KDM4E (0.46) KDM4EALDH1A1USP2MAPTCYP19A1
SCHEMBL8540882 0.76 AR (0.43) ALDH1A1USP2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100534987-C New method for preparing 2-methoxy-5(5-trifluoromethyl-1H-tetraazo-1-group) benzaldehyde CHENGDU MOLECULAR LAB CO LTD (CN) 2009-09-02 CN disclosed
CN-1882345-A 2, 6-disubstituted quinazolines, quinoxalines, quinolines and isoquinolines as RAF kinase inhibitors for the treatment of cancer CHIRON CORP (US) 2006-12-20 CN disclosed
CN-1850810-A New method for preparing 2-methoxy-5(5-trifluoromethyl-1H-tetraazo-1-group) benzaldehyde CHENGDU MOLECULAR LAB CO LTD (CN) 2006-10-25 CN disclosed
EP-0665843-B1 SUBSTITUTED QUINUCLIDINES AS SUBSTANCE P ANTAGONISTS PFIZER (US) 2003-08-13 EP disclosed
US-5837711-A Substituted quinuclidines as substance P antagonists PFIZER INC. (US) 1998-11-17 US disclosed
EP-0665843-A1 SUBSTITUTED QUINUCLIDINES AS SUBSTANCE P ANTAGONISTS PFIZER INC. (US) 1995-08-09 EP disclosed
WO-1994010170-A1 SUBSTITUTED QUINUCLIDINES AS SUBSTANCE P ANTAGONISTS PFIZER INC. (US) 1994-05-11 WO disclosed