SCHEMBL7819793

SCHEMBL7819793

Nc1ccc(OC(F)(F)F)c(C2OCCO2)c1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.31
BACE1 P56817 1/20 0.31
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
GLA P06280 1/20 0.30
POLB P06746 1/20 0.30
GAA P10253 1/20 0.30
TSHR P16473 1/20 0.30
PDE2A O00408 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30975319 0.81 SLC6A4 (0.34) GRIN2B
SCHEMBL7090123 0.79 KDM4E (0.42) GAATSHR
SCHEMBL25468145 0.79 CHRNB2 (0.35) GRIN2BHCRTR1HCRTR2GLAPOLB
SCHEMBL7811713 0.76 AKR1C3 (0.39)
SCHEMBL22816076 0.74 PDE10A (0.32) BACE1
SCHEMBL21962283 0.73 KDM1A (0.35) BACE1GAA
SCHEMBL7818101 0.73 KIF11 (0.46)
SCHEMBL7234652 0.72 MEN1 (0.33)
SCHEMBL12952676 0.72 RAB9A (0.50) POLB
SCHEMBL9367414 0.72 GAA (0.40) GLAPOLBGAATSHRPDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0655996-B1 SUBSTITUTED BENZYLAMINO NITROGEN CONTAINING NON-AROMATIC HETEROCYCLES PFIZER (US) 2001-11-07 EP disclosed
EP-1114823-A2 Substituted benzylamino nitrogen containing non-aromatic heterocycles PFIZER INC. (US) 2001-07-11 EP disclosed
US-5721255-A Substituted benzylamino nitrogen containing non-aromatic heterocycles PFIZER INC. (US) 1998-02-24 US disclosed