SCHEMBL7090430

SCHEMBL7090430

Clc1cccc(Cl)c1CSc1nnc(-c2ccccc2)n1Cc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.56
MEN1 O00255 4/20 0.54
KMT2A Q03164 4/20 0.54
CYP3A4 P08684 2/20 0.54
CYP2C19 P33261 2/20 0.54
CYP1A2 P05177 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
ALDH1A1 P00352 4/20 0.54
HTT P42858 3/20 0.54
LMNA P02545 4/20 0.53
SMN1; SMN2 Q16637 6/20 0.52
TSHR P16473 4/20 0.52
NPC1 O15118 2/20 0.52
RAB9A P51151 1/20 0.52
GAA P10253 2/20 0.51
OPRK1 P41145 2/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3915525 0.86 ALDH1A1 (0.67) KDM4EMEN1KMT2ACYP3A4CYP2C19
SCHEMBL3910599 0.83 ALDH1A1 (0.60) KDM4EMEN1KMT2ACYP3A4CYP2C19
SCHEMBL4211347 0.78 TSHR (0.56) MEN1KMT2ACYP3A4CYP2C19CYP1A2
SCHEMBL6402415 0.77 ALDH1A1 (0.74) KDM4EALDH1A1LMNASMN1; SMN2TSHR
SCHEMBL6410240 0.77 MEN1 (0.70) KDM4EMEN1KMT2ACYP3A4CYP2C19
SCHEMBL3904873 0.76 TSHR (0.67) KDM4EMEN1KMT2ACYP3A4ALDH1A1
SCHEMBL4218132 0.76 ALDH1A1 (0.63) KDM4EMEN1KMT2AALDH1A1HTT
SCHEMBL15983422 0.75 ALDH1A1 (0.80) KDM4EMEN1KMT2AALDH1A1LMNA
SCHEMBL4204703 0.74 SMN1; SMN2 (0.61) CYP3A4CYP2C19CYP1A2CYP2C9ALDH1A1
SCHEMBL4215484 0.74 ALDH1A1 (0.69) KDM4EMEN1KMT2ACYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1357913-A1 HETEROCYCLIC INHIBITORS OF GLYCINE TRANSPORTER 2 TELIK, INC. (US) 2003-11-05 EP claimed
WO-2002064135-A1 HETEROCYCLIC INHIBITORS OF GLYCINE TRANSPORTER 2 TELIK, INC. (US) 2002-08-22 WO claimed
EP-1357913-A1 HETEROCYCLIC INHIBITORS OF GLYCINE TRANSPORTER 2 TELIK, INC. (US) 2003-11-05 EP disclosed
WO-2002064135-A1 HETEROCYCLIC INHIBITORS OF GLYCINE TRANSPORTER 2 TELIK, INC. (US) 2002-08-22 WO disclosed