SCHEMBL7092448

SCHEMBL7092448

c1nc(OCCN2CCCCC2)cc2c1CCN2

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 12/20 0.52
LTA4H P09960 2/20 0.42
HRH1 P35367 1/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNA4 P43681 1/20 0.41
SLC6A4 P31645 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
PTGS2 P35354 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7094573 0.77 HRH3 (0.77) HRH3HRH1
SCHEMBL15897912 0.76 HRH3 (0.74) HRH3LTA4HHRH1
SCHEMBL7094592 0.75 HRH3 (0.54) HRH3LTA4HHRH1
SCHEMBL7096511 0.75 HRH3 (0.54) HRH3HRH1
SCHEMBL7097649 0.74 EHMT2 (0.55) HRH3LTA4H
Hydrochloric Acid SCHEMBL6109241 0.74 HRH3 (0.85) HRH3LTA4HHRH1
SCHEMBL7094760 0.73 HRH3 (0.52) HRH3HRH1
SCHEMBL7092953 0.73 EHMT2 (0.56) HRH3LTA4H
SCHEMBL7094490 0.73 HRH3 (0.51) HRH3HRH1
SCHEMBL7094945 0.73 HRH3 (0.51) HRH3LTA4HHRH1HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1309551-A1 INDOLINE DERIVATIVES AS 5HT2C ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 2003-05-14 EP disclosed
WO-2002014273-A1 INDOLINE DERIVATIVES AS 5HT2C ANTAGONISTS SMITHKLINE BEECHAM P.L.C. (GB) 2002-02-21 WO disclosed