SCHEMBL7092816

SCHEMBL7092816

COc1ccc(-c2sc3cc(OC)ccc3c2-c2cc(OCCN3CCCCC3)ccc2C=O)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 13/20 0.63
ESR2 Q92731 13/20 0.63
ENPP3 O14638 3/20 0.53
ENPP1 P22413 2/20 0.53
UBE2N P61088 1/20 0.49
ITGA4 P13612 1/20 0.49
MEN1 O00255 1/20 0.48
PLD2 O14939 1/20 0.48
KDM1A O60341 1/20 0.48
NR1I2 O75469 1/20 0.48
USP2 O75604 1/20 0.48
ALDH1A1 P00352 1/20 0.48
C5 P01031 1/20 0.48
LMNA P02545 1/20 0.48
TP53 P04637 1/20 0.48
FYN P06241 1/20 0.48
PGR P06401 1/20 0.48
CYP3A4 P08684 1/20 0.48
ADRA2A P08913 1/20 0.48
ADORA3 P0DMS8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL987943 0.88 ESR1 (0.64) ESR1ESR2UBE2NMEN1PLD2
Hydrochloric Acid SCHEMBL8866853 0.88 ENPP3 (0.56) ESR1ESR2ENPP3ENPP1UBE2N
Hydrochloric Acid SCHEMBL3974968 0.87 ESR1 (0.64) ESR1ESR2UBE2NMEN1PLD2
SCHEMBL5409936 0.84 TUBB4A (0.47) ESR1ESR2ALDH1A1MAPTCNR1
SCHEMBL7942841 0.82 ESR1 (0.52) ESR1ESR2ENPP3ENPP1ITGA4
SCHEMBL7944330 0.82 ESR1 (0.51) ESR1ESR2ENPP3ENPP1ITGA4
SCHEMBL7944288 0.82 ESR1 (0.51) ESR1ESR2ENPP3ENPP1ITGA4
Hydrochloric Acid SCHEMBL7100412 0.82 ESR1 (0.66) ESR1ESR2ENPP3ENPP1UBE2N
Hydrochloric Acid SCHEMBL7097572 0.81 ESR1 (0.64) ESR1ESR2ENPP3ENPP1UBE2N
SCHEMBL6749914 0.81 BCHE (0.58) ESR1ESR2ALDH1A1MAPTACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0979076-A4 INTERMEDIATES AND PROCESSES FOR PREPARING BENZO b]THIOPHENES LILLY CO ELI (US) 2003-03-19 EP disclosed
EP-0979076-A1 INTERMEDIATES AND PROCESSES FOR PREPARING BENZO b]THIOPHENES ELI LILLY AND COMPANY (US) 2000-02-16 EP disclosed
US-6018056-A Intermediates and processes for preparing benzo (b) thiophenes ELI LILLY AND COMPANY (US) 2000-01-25 US disclosed
WO-1998048793-A1 INTERMEDIATES AND PROCESSES FOR PREPARING BENZO[b]THIOPHENES ELI LILLY AND COMPANY (US) 1998-11-05 WO disclosed