SCHEMBL7092828

SCHEMBL7092828

O=c1[nH]c(=S)[nH]c(-c2ccc(Cl)cc2)c1-c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.55
HSD17B10 Q99714 2/20 0.55
HPGD P15428 1/20 0.55
TYMP P19971 1/20 0.46
SERPINE1 P05121 1/20 0.45
KDM4E B2RXH2 1/20 0.43
MDM2 Q00987 1/20 0.43
CYP1A2 P05177 2/20 0.42
PTGS2 P35354 4/20 0.42
LMNA P02545 2/20 0.41
GSK3B P49841 2/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
ROCK2 O75116 1/20 0.40
MAP4K4 O95819 1/20 0.40
LCK P06239 1/20 0.40
CSF1R P07333 1/20 0.40
PIM1 P11309 1/20 0.40
RPS6KB1 P23443 1/20 0.40
CDK2 P24941 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7093919 1.00 ALDH1A1 (0.55) ALDH1A1HSD17B10HPGDTYMPSERPINE1
SCHEMBL7090889 0.90 HSD17B10 (0.66) ALDH1A1HSD17B10HPGDTYMPSERPINE1
SCHEMBL7089988 0.86 POLB (0.55) ALDH1A1HSD17B10HPGDSERPINE1MDM2
SCHEMBL7091477 0.84 POLB (0.56) ALDH1A1HSD17B10HPGDTYMPMDM2
SCHEMBL1573392 0.84 TYMP (0.62) ALDH1A1HSD17B10HPGDTYMPSERPINE1
SCHEMBL1573566 0.84 TYMP (0.62) ALDH1A1HSD17B10HPGDTYMPSERPINE1
SCHEMBL7093329 0.81 HSD17B10 (0.51) ALDH1A1HSD17B10HPGDTYMPMDM2
SCHEMBL7094140 0.81 ALDH1A1 (0.51) ALDH1A1HSD17B10HPGDTYMPMDM2
SCHEMBL7093922 0.81 ALDH1A1 (0.51) ALDH1A1HSD17B10HPGDKDM4EMDM2
SCHEMBL7092623 0.80 PTGS2 (0.60) ALDH1A1HSD17B10HPGDPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003084935-A2 DIARYL PYRIMIDINONE DERIVATIVES USEFUL FOR THE TREATMENT OF INFLAMMATION AND IMMUNOGOLICAL DISEASES ORCHID CHEMICALS & PHARMACEUTICALS LTD (IN) 2003-10-16 WO claimed
WO-2003084935-A2 DIARYL PYRIMIDINONE DERIVATIVES USEFUL FOR THE TREATMENT OF INFLAMMATION AND IMMUNOGOLICAL DISEASES ORCHID CHEMICALS & PHARMACEUTICALS LTD (IN) 2003-10-16 WO disclosed