SCHEMBL7093329

SCHEMBL7093329

CSc1ccc(-c2c(-c3ccccc3)[nH]c(=S)[nH]c2=O)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.51
ALDH1A1 P00352 1/20 0.51
HPGD P15428 1/20 0.51
PTGS2 P35354 3/20 0.48
MDM2 Q00987 1/20 0.44
GSK3B P49841 1/20 0.41
POLB P06746 1/20 0.40
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38
CYP2C19 P33261 1/20 0.38
HIF1A Q16665 1/20 0.38
SIRT2 Q8IXJ6 1/20 0.38
SIRT1 Q96EB6 1/20 0.38
SIRT3 Q9NTG7 1/20 0.38
SIRT5 Q9NXA8 1/20 0.38
SMPD3 Q9NY59 1/20 0.38
XDH P47989 1/20 0.38
PTGS1 P23219 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7090889 0.86 HSD17B10 (0.66) HSD17B10ALDH1A1HPGDMDM2POLB
SCHEMBL1573106 0.85 PTGS2 (0.50) HSD17B10ALDH1A1HPGDPTGS2MDM2
SCHEMBL7091477 0.84 POLB (0.56) HSD17B10ALDH1A1HPGDPTGS2MDM2
SCHEMBL7092828 0.81 ALDH1A1 (0.55) HSD17B10ALDH1A1HPGDPTGS2MDM2
SCHEMBL7093919 0.81 ALDH1A1 (0.55) HSD17B10ALDH1A1HPGDPTGS2MDM2
SCHEMBL7093922 0.80 ALDH1A1 (0.51) HSD17B10ALDH1A1HPGDPTGS2MDM2
SCHEMBL7092623 0.79 PTGS2 (0.60) HSD17B10ALDH1A1HPGDPTGS2PTGS1
SCHEMBL11186325 0.78 PTGS2 (0.39) ALDH1A1PTGS2GSK3BPOLB
SCHEMBL7094140 0.77 ALDH1A1 (0.51) HSD17B10ALDH1A1HPGDMDM2CYP1A2
SCHEMBL7090564 0.76 PTGS2 (0.60) HSD17B10ALDH1A1HPGDPTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003084935-A2 DIARYL PYRIMIDINONE DERIVATIVES USEFUL FOR THE TREATMENT OF INFLAMMATION AND IMMUNOGOLICAL DISEASES ORCHID CHEMICALS & PHARMACEUTICALS LTD (IN) 2003-10-16 WO claimed
WO-2003084935-A2 DIARYL PYRIMIDINONE DERIVATIVES USEFUL FOR THE TREATMENT OF INFLAMMATION AND IMMUNOGOLICAL DISEASES ORCHID CHEMICALS & PHARMACEUTICALS LTD (IN) 2003-10-16 WO disclosed