SCHEMBL7093772

SCHEMBL7093772

NC(=O)c1ccccc1N(c1ccccc1)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.47
ALDH1A1 P00352 7/20 0.47
MAPT P10636 5/20 0.47
TSHR P16473 4/20 0.47
KDM4E B2RXH2 4/20 0.47
HSD17B10 Q99714 2/20 0.47
HPGD P15428 2/20 0.47
METAP2 P50579 1/20 0.44
CTNNB1 P35222 1/20 0.43
SIRT1 Q96EB6 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
CYP3A4 P08684 2/20 0.41
CYP2C19 P33261 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
POLB P06746 1/20 0.41
PARP1 P09874 1/20 0.41
RECQL P46063 1/20 0.41
BLM P54132 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28734017 0.85 BCAT2 (0.42) BCAT2ALDH1A1MAPTTSHRKDM4E
SCHEMBL1227194 0.83 ALDH1A1 (0.54) ALDH1A1MAPTTSHRKDM4EHPGD
SCHEMBL27863652 0.83 BCAT2 (0.47) BCAT2ALDH1A1MAPTTSHRKDM4E
SCHEMBL10992096 0.82 SIRT1 (0.46) BCAT2ALDH1A1MAPTTSHRKDM4E
SCHEMBL2762268 0.81 MAPT (0.46) BCAT2ALDH1A1MAPTTSHRKDM4E
SCHEMBL3644388 0.81 NPSR1 (0.47) BCAT2ALDH1A1MAPTTSHRKDM4E
SCHEMBL7259310 0.80 ALDH1A1 (0.44) BCAT2ALDH1A1MAPTTSHRKDM4E
SCHEMBL31179917 0.80 ALDH1A1 (0.44) ALDH1A1MAPTTSHRKDM4EPOLB
SCHEMBL13587852 0.79 ALDH1A1 (0.54) ALDH1A1MAPTTSHRKDM4EHPGD
SCHEMBL21808781 0.78 AKR1C3 (0.53) ALDH1A1MAPTTSHRKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003082777-A2 NOVEL GLUCOCORTICOID RECEPTOR LIGANDS KARO BIO AB (SE) 2003-10-09 WO claimed
WO-2003082777-A2 NOVEL GLUCOCORTICOID RECEPTOR LIGANDS KARO BIO AB (SE) 2003-10-09 WO disclosed