Formamide

Formamide

SCHEMBL7094949

NC=O.NCCc1ccc(NC2CCN(C(=O)NCc3cc(F)cc(F)c3)CC2)cc1

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 9/20 0.51
ADRB1 P08588 8/20 0.51
ADRB2 P07550 1/20 0.46
TPSAB1 Q15661 2/20 0.43
TPSD1 Q9BZJ3 2/20 0.43
TPSG1 Q9NRR2 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ALDH1A1 P00352 1/20 0.43
TSHR P16473 1/20 0.43
MLNR O43193 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Formic Acid SCHEMBL7097395 0.96 ADRB3 (0.51) ADRB3ADRB1ADRB2TPSAB1TPSD1
Formic Acid SCHEMBL7094256 0.88 ADRB1 (0.59) ADRB3ADRB1ADRB2TPSAB1TPSD1
Formic Acid SCHEMBL7094276 0.87 ADRB3 (0.49) ADRB3ADRB1ADRB2MEN1KMT2A
SCHEMBL7094555 0.87 ADRB1 (0.60) ADRB3ADRB1ADRB2TPSAB1TPSD1
SCHEMBL7092013 0.85 ADRB3 (0.53) ADRB3ADRB1ADRB2TPSAB1MEN1
Formic Acid SCHEMBL7094738 0.83 ADRB3 (0.63) ADRB3ADRB1ADRB2TPSAB1TPSD1
Formic Acid SCHEMBL7096875 0.83 ADRB1 (0.63) ADRB3ADRB1ADRB2TPSAB1TPSD1
SCHEMBL7094506 0.83 ADRB1 (0.64) ADRB3ADRB1ADRB2TPSAB1TPSD1
Formic Acid SCHEMBL7096141 0.82 ADRB3 (0.61) ADRB3ADRB1ADRB2TPSAB1TPSD1
Formic Acid SCHEMBL7095380 0.82 TPSAB1 (0.57) ADRB3ADRB1ADRB2TPSAB1TPSD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6605618-B2 Antidiabetic agents; hypoglycemic agents; anticholesterol agents; side effect reduction WYETH 2003-08-12 US disclosed
US-20030018045-A1 Heterocyclic beta-3 adrenergic receptor agonists WYETH (US) 2003-01-23 US disclosed
US-6451814-B1 SUBSTITUTED 4-((4-AMINO-5-HYDROXYPHENYL)-OXY-)PIPERIDINE ANALOGS; METABOLIC DISORDERS; ANTIDIABETIC AGENTS; ATHERO-SCLEROSIS, GASTROINTESTINAL DISORDERS, GLAUCOMA, NEUROGENETIC INFLAMMATION, OCULAR HYPERTENSION AND FREQUENT URINATION WYETH 2002-09-17 US disclosed
US-20020028832-A1 Heterocyclic beta-3 adrenergic receptor agonists AMERICAN HOME PRODUCTS CORPORATION (US) 2002-03-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030018045-A1 Heterocyclic beta-3 adrenergic receptor agonists ADRB2, ADRB1, ADRB3 ADRB3 3/4885ADRB1 2/4885ADRB2 1/4885
US-20020028832-A1 Heterocyclic beta-3 adrenergic receptor agonists ADRB1, ADRB3, ADRB2 ADRB3 2/4885ADRB1 1/4885ADRB2 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.