SCHEMBL7095155

SCHEMBL7095155

O=c1[nH]c(-c2ccc(C(F)(F)F)cc2)c(-c2ccccc2)c(=O)[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMP P19971 4/20 0.53
GAA P10253 2/20 0.50
ALDH1A1 P00352 2/20 0.50
KDM4E B2RXH2 1/20 0.50
PLA2G10 O15496 1/20 0.50
HPGD P15428 1/20 0.50
HSD17B10 Q99714 1/20 0.50
KIF11 P52732 1/20 0.50
BACE1 P56817 1/20 0.47
TNKS O95271 1/20 0.46
WNT3A P56704 1/20 0.46
TNKS2 Q9H2K2 1/20 0.46
MAPK13 O15264 1/20 0.44
RAF1 P04049 1/20 0.44
MAPK12 P53778 1/20 0.44
MAPK11 Q15759 1/20 0.44
MAPK14 Q16539 1/20 0.44
SCN2A Q99250 2/20 0.42
MGAM O43451 1/20 0.41
SI P14410 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7094140 0.85 ALDH1A1 (0.51) TYMPGAAALDH1A1HPGDHSD17B10
SCHEMBL1572915 0.85 ALDH1A1 (0.68) TYMPGAAALDH1A1KDM4EPLA2G10
SCHEMBL30472340 0.81 TNKS (0.55) GAAKIF11BACE1TNKSWNT3A
SCHEMBL29031843 0.81 TNKS (0.55) GAAKIF11BACE1TNKSWNT3A
SCHEMBL8354646 0.80 MAPK14 (0.53) GAAALDH1A1KDM4EPLA2G10HPGD
SCHEMBL1573566 0.80 TYMP (0.62) TYMPGAAALDH1A1KDM4EPLA2G10
SCHEMBL1573105 0.80 KDM4E (0.55) TYMPGAAALDH1A1KDM4EPLA2G10
SCHEMBL1573392 0.80 TYMP (0.62) TYMPGAAALDH1A1KDM4EPLA2G10
SCHEMBL1573106 0.76 PTGS2 (0.50) TYMPGAAALDH1A1KDM4EPLA2G10
SCHEMBL1573422 0.76 KDM4E (0.50) TYMPGAAALDH1A1KDM4EPLA2G10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003084935-A2 DIARYL PYRIMIDINONE DERIVATIVES USEFUL FOR THE TREATMENT OF INFLAMMATION AND IMMUNOGOLICAL DISEASES ORCHID CHEMICALS & PHARMACEUTICALS LTD (IN) 2003-10-16 WO claimed
WO-2003084935-A2 DIARYL PYRIMIDINONE DERIVATIVES USEFUL FOR THE TREATMENT OF INFLAMMATION AND IMMUNOGOLICAL DISEASES ORCHID CHEMICALS & PHARMACEUTICALS LTD (IN) 2003-10-16 WO disclosed