SCHEMBL7095601

SCHEMBL7095601

Nc1c[c]cc(C(=O)NCCCc2ccccc2)c1

nearest known ligand 0.62

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.62
RAB9A P51151 3/20 0.62
POLB P06746 2/20 0.61
KDM4E B2RXH2 1/20 0.61
SMN1; SMN2 Q16637 2/20 0.52
MLYCD O95822 1/20 0.52
EPHX2 P34913 1/20 0.52
HSP90AA1 P07900 1/20 0.51
HPGD P15428 3/20 0.51
ALDH1A1 P00352 2/20 0.51
GPR84 Q9NQS5 1/20 0.50
MAPT P10636 1/20 0.50
TSHR P16473 1/20 0.50
HTT P42858 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
HSD17B10 Q99714 1/20 0.50
NLRP1 Q9C000 1/20 0.50
PKM P14618 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5847828 0.83 HDAC6 (0.53) RAB9ASMN1; SMN2HPGDALDH1A1TSHR
SCHEMBL5847797 0.79 ALDH1A1 (0.47) NPC1RAB9APOLBKDM4ESMN1; SMN2
SCHEMBL3225126 0.78 NPC1 (1.00) NPC1RAB9APOLBKDM4ESMN1; SMN2
Hydrochloric Acid SCHEMBL6961822 0.77 NPC1 (0.64) NPC1RAB9APOLBKDM4ESMN1; SMN2
SCHEMBL2956025 0.77 NPC1 (0.68) NPC1RAB9APOLBKDM4ESMN1; SMN2
SCHEMBL7105034 0.76 LMNA (0.57) NPC1RAB9AKDM4ESMN1; SMN2MAPT
SCHEMBL6240951 0.76 L3MBTL1 (0.46) POLBKDM4ESMN1; SMN2HPGDALDH1A1
SCHEMBL8476710 0.76 NPC1 (0.66) NPC1RAB9APOLBKDM4ESMN1; SMN2
SCHEMBL4930583 0.75 NPC1 (0.64) NPC1RAB9APOLBKDM4ESMN1; SMN2
SCHEMBL4628943 0.74 NPC1 (0.68) NPC1RAB9APOLBKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001087852-A1 SUBSTITUTED POLYCYCLIC ARYL AND HETEROARYL URACILS USEFUL FOR SELECTIVE INHIBITION OF THE COAGULATION CASCADE PHARMACIA CORPORATION (US) 2001-11-22 WO claimed
EP-1268428-A2 POLYCYCLIC ARYL AND HETEROARYL SUBSTITUTED 4-PYRIDONES USEFUL FOR SELECTIVE INHIBITION OF THE COAGULATION CASCADE Pharmacia Corporation (US) 2003-01-02 EP disclosed
WO-2001077079-A2 POLYCYCLIC ARYL AND HETEROARYL SUBSTITUTED 4-PYRIDONES USEFUL FOR SELECTIVE INHIBITION OF THE COAGULATION CASCADE PHARMACIA CORPORATION (US) 2001-10-18 WO disclosed