SCHEMBL7095832

SCHEMBL7095832

c1ccc2c(c1)sc1c(-c3ccc(CNc4ccc(OCCN5CCOCC5)nc4)cc3)n[nH]c12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 8/20 0.40
UBE2N P61088 1/20 0.40
ABL1 P00519 1/20 0.39
TUBB4A P04350 1/20 0.39
TUBB P07437 1/20 0.39
LYN P07948 1/20 0.39
TUBA3C P0DPH7 1/20 0.39
BCR P11274 1/20 0.39
SRC P12931 1/20 0.39
TUBA1B P68363 1/20 0.39
TUBA4A P68366 1/20 0.39
TUBB4B P68371 1/20 0.39
TUBB3 Q13509 1/20 0.39
TUBB2A Q13885 1/20 0.39
TUBB8 Q3ZCM7 1/20 0.39
TUBA3E Q6PEY2 1/20 0.39
TUBA1A Q71U36 1/20 0.39
TUBA1C Q9BQE3 1/20 0.39
TUBB6 Q9BUF5 1/20 0.39
TUBB2B Q9BVA1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7093132 0.82 HTR6 (0.37) KDRTLR7
SCHEMBL6998526 0.81 PARP1 (0.47) MEN1KMT2AALDH1A1LMNAKDM4E
Hydrochloric Acid SCHEMBL7006248 0.80 PARP1 (0.46) MEN1KMT2AALDH1A1LMNAKDM4E
SCHEMBL7097405 0.77 KDM4E (0.41) AURKBABL1SRCKMT2AALDH1A1
SCHEMBL7094580 0.73 RAB9A (0.46) KDM4ELTA4H
SCHEMBL7090927 0.72 GAA (0.46) MEN1KMT2AHIF1AKDM4EMAPT
SCHEMBL7096045 0.72 LRRK2 (0.43) AURKBLYNF2FLT3
SCHEMBL7094609 0.70 NTRK1 (0.43) AURKA
SCHEMBL7092191 0.69 CXCR4 (0.51) AURKBABL1SRCMEN1KMT2A
SCHEMBL5872943 0.67 ALDH1A1 (0.43) UBE2NMEN1KMT2AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268437-A1 INHIBITORS OF PROTEIN KINASES Knoll GmbH (DE) 2003-01-02 EP disclosed
WO-2002030908-A1 INHIBITORS OF PROTEIN KINASES KNOLL GMBH (DE) 2002-04-18 WO disclosed
US-6297238-B1 3-ARYL PYRAZOLES WITH 4,5(3,4)-BICYCLIC RING FUSION WHICH ARE INHIBITORS OF PROTEIN KINASES PARTICULARLY TYROSINE KINASES AND SERINE/THREONINE KINASES BASF AKTIENGESELLSCHAFT (DE) 2001-10-02 US disclosed