SCHEMBL7096028

SCHEMBL7096028

Cc1c(S(=O)(=O)n2ccc(C3CCCNC3)c2)sc2ccc(Cl)cc12

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 17/20 0.66
NPSR1 Q6W5P4 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HTR1A P08908 4/20 0.40
HTR1D P28221 4/20 0.40
HTR1B P28222 4/20 0.40
HTR2C P28335 3/20 0.40
DRD2 P14416 2/20 0.40
HTR7 P34969 2/20 0.40
ADRA1B P35368 2/20 0.40
DRD3 P35462 2/20 0.40
HTR4 Q13639 2/20 0.40
DRD1 P21728 1/20 0.40
DRD4 P21917 1/20 0.40
HTR2A P28223 1/20 0.40
AKR1B1 P15121 1/20 0.40
CYP1A2 P05177 1/20 0.39
ADRB1 P08588 1/20 0.39
CYP3A4 P08684 1/20 0.39
ADRA2A P08913 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5255669 0.79 HTR6 (1.00) HTR6HTR1A
SCHEMBL5252115 0.77 HTR6 (0.77) HTR6HTR1AHTR1DHTR1B
SCHEMBL13598936 0.67 HTR6 (0.58) HTR6NPSR1L3MBTL1HTR1AHTR1D
SCHEMBL7103771 0.67 HTR6 (0.45) HTR6L3MBTL1HTR2ACYP2D6SLC6A2
SCHEMBL7164227 0.66 PKM (0.47) HTR6SLC6A2
SCHEMBL4427807 0.65 HTR6 (0.53) HTR6NPSR1L3MBTL1HTR1AHTR1D
SCHEMBL13696908 0.65 NPSR1 (0.62) HTR6NPSR1L3MBTL1AKR1B1
SCHEMBL1548591 0.65 NPSR1 (0.62) HTR6NPSR1L3MBTL1AKR1B1
SCHEMBL337593 0.65 NPSR1 (0.62) NPSR1L3MBTL1AKR1B1
SCHEMBL3681454 0.65 NPSR1 (0.59) HTR6NPSR1L3MBTL1DRD2HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355904-A2 HETEROCYCLINDAZOLE AND AZAINDAZOLE COMPOUNDS AS 5-HYDROXYTRYPTAMINE-6 LIGANDS Wyeth (US) 2003-10-29 EP claimed
WO-2002051837-A2 HETEROCYCLINDAZOLE AND AZAINDAZOLE COMPOUNDS AS 5-HYDROXYTRYPTAMINE-6 LIGANDS WYETH (US) 2002-07-04 WO claimed