SCHEMBL7096838

SCHEMBL7096838

COP(=O)(CCn1c(=O)[nH]c(=O)c2c1ncn2C)OC

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 5/20 0.65
ADORA2A P29274 5/20 0.65
PDE4B Q07343 5/20 0.65
PDE4C Q08493 5/20 0.65
PDE4D Q08499 5/20 0.65
CYP3A4 P08684 2/20 0.54
PMP22 Q01453 2/20 0.54
MAPK1 P28482 1/20 0.54
MEN1 O00255 1/20 0.48
ALDH1A1 P00352 1/20 0.48
KMT2A Q03164 1/20 0.48
BRD4 O60885 4/20 0.47
BRD2 P25440 2/20 0.47
BRD3 Q15059 2/20 0.47
BRDT Q58F21 2/20 0.47
ADORA2B P29275 3/20 0.39
CYP1A2 P05177 1/20 0.39
BLM P54132 1/20 0.39
HSD17B10 Q99714 1/20 0.39
GDA Q9Y2T3 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7101360 0.80 BLM (0.54) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL12257284 0.78 PDE4A (0.80) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL10813831 0.77 PDE4A (0.83) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL10571805 0.76 PDE4A (0.78) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL7099928 0.76 ADORA2B (0.50) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL7781761 0.76 KDM4E (0.39) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL29474230 0.75 PDE4A (0.70) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL2462137 0.74 PDE4A (0.69) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL7100345 0.73 ADORA2B (0.50) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL32679497 0.73 PDE4A (0.68) PDE4AADORA2APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140952-B1 ORGANO-PHOSPHORUS COMPOUNDS AND THEIR UTILIZATION BIOAGENCY AG (DE) 2003-09-03 EP disclosed
EP-1140952-A1 ORGANO-PHOSPHORUS COMPOUNDS AND THEIR UTILIZATION Jomaa Pharmaka GmbH (DE) 2001-10-10 EP disclosed
WO-2000037477-A1 ORGANO-PHOSPHORUS COMPOUNDS AND THEIR UTILIZATION JOMAA PHARMAKA GMBH (DE) 2000-06-29 WO disclosed