SCHEMBL7100345

SCHEMBL7100345

COP(=O)(CCn1c(=O)c2c(ncn2C)n(O)c1=O)OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 8/20 0.50
PDE4A P27815 4/20 0.50
PDE4B Q07343 4/20 0.50
PDE4C Q08493 4/20 0.50
PDE4D Q08499 4/20 0.50
ADORA2A P29274 3/20 0.50
BLM P54132 2/20 0.50
CYP1A2 P05177 2/20 0.50
PMP22 Q01453 2/20 0.50
CYP3A4 P08684 1/20 0.50
HSD17B10 Q99714 1/20 0.50
TNF P01375 3/20 0.46
GLA P06280 1/20 0.45
USP2 O75604 1/20 0.44
LMNA P02545 1/20 0.44
TSHR P16473 1/20 0.44
NFKB1 P19838 1/20 0.44
ACHE P22303 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7099928 0.90 ADORA2B (0.50) ADORA2BPDE4APDE4BPDE4CPDE4D
SCHEMBL7100798 0.76 ADORA2B (0.55) ADORA2BPDE4APDE4BPDE4CPDE4D
SCHEMBL7096838 0.73 PDE4A (0.65) ADORA2BPDE4APDE4BPDE4CPDE4D
SCHEMBL7101360 0.73 BLM (0.54) ADORA2BPDE4APDE4BPDE4CPDE4D
SCHEMBL7460040 0.69 TNF (0.63) ADORA2BPDE4APDE4BPDE4CPDE4D
Bisdionin B SCHEMBL29896692 0.69 ADORA2B (0.74) ADORA2BPDE4APDE4BPDE4CPDE4D
SCHEMBL7464356 0.68 TNF (0.64) ADORA2BPDE4APDE4BPDE4CPDE4D
SCHEMBL8658922 0.68 ADORA2B (0.63) ADORA2BPDE4APDE4BPDE4CPDE4D
SCHEMBL316911 0.68 PDE4A (1.00) ADORA2BPDE4APDE4BPDE4CPDE4D
SCHEMBL7459098 0.68 TNF (0.62) ADORA2BPDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140952-B1 ORGANO-PHOSPHORUS COMPOUNDS AND THEIR UTILIZATION BIOAGENCY AG (DE) 2003-09-03 EP disclosed
EP-1140952-A1 ORGANO-PHOSPHORUS COMPOUNDS AND THEIR UTILIZATION Jomaa Pharmaka GmbH (DE) 2001-10-10 EP disclosed
WO-2000037477-A1 ORGANO-PHOSPHORUS COMPOUNDS AND THEIR UTILIZATION JOMAA PHARMAKA GMBH (DE) 2000-06-29 WO disclosed