SCHEMBL7097552

SCHEMBL7097552

CNN1CCCCCC1c1cncc(F)c1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.42
JAK2 O60674 9/20 0.41
NTRK1 P04629 9/20 0.41
CHRNA1 P02708 1/20 0.37
CHRNG P07510 1/20 0.37
CHRNB1 P11230 1/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA4 P43681 1/20 0.37
CHRND Q07001 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7098412 0.99 RIPK1 (0.43) RIPK1JAK2NTRK1CHRNA1CHRNG
SCHEMBL7101650 0.94 JAK2 (0.45) RIPK1JAK2NTRK1CHRNA1CHRNG
SCHEMBL7097804 0.81 KDM4E (0.40) CHRNA1CHRNGCHRNB1CHRNB2CHRNB4
SCHEMBL7097799 0.80 CHRNB4 (0.46) CHRNA1CHRNGCHRNB1CHRNB2CHRNB4
SCHEMBL7099484 0.80 CHRNA3 (0.62) CHRNA1CHRNGCHRNB1CHRNB2CHRNB4
SCHEMBL7101914 0.80 KDM4E (0.41) CHRNA1CHRNGCHRNB1CHRNB2CHRNB4
SCHEMBL7098421 0.78 CHRNB4 (0.47) CHRNA1CHRNGCHRNB1CHRNB2CHRNB4
SCHEMBL7101829 0.78 CHRNA3 (0.64) CHRNA1CHRNGCHRNB1CHRNB2CHRNB4
SCHEMBL7100521 0.77 OPRK1 (0.31)
SCHEMBL7098886 0.77 KMT2A (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003500402-A 2003-01-07 JP claimed
EP-1178982-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2002-02-13 EP claimed
WO-2000071534-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2000-11-30 WO claimed
EP-1178982-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2002-02-13 EP disclosed
WO-2000071534-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2000-11-30 WO disclosed