SCHEMBL7097607

SCHEMBL7097607

O=C(O)Cn1c(=O)n(Cc2ccccc2)c(=O)c2cc(C(=O)NCc3ccc4c(c3)OCO4)ccc21

nearest known ligand 0.69

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPT P10636 10/20 0.68
POLB P06746 4/20 0.66
TP53 P04637 3/20 0.65
THRB P10828 1/20 0.65
TDP1 Q9NUW8 1/20 0.65
KMT2A Q03164 2/20 0.62
MEN1 O00255 1/20 0.62
USP2 O75604 1/20 0.62
PPARG P37231 2/20 0.58
HTT P42858 1/20 0.55
ESR1 P03372 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27605963 0.88 MAPT (0.61) MAPTPOLBTP53THRBTDP1
SCHEMBL7171065 0.86 MAPT (0.57) MAPTPOLBTP53THRBTDP1
SCHEMBL6259247 0.83 PPARG (0.57) MAPTPOLBTP53THRBTDP1
SCHEMBL7622582 0.82 USP2 (0.61) MAPTTP53KMT2AMEN1USP2
SCHEMBL6210665 0.82 PPARG (0.54) MAPTPOLBTP53THRBTDP1
SCHEMBL6213391 0.82 PPARG (0.54) MAPTPOLBTP53THRBTDP1
SCHEMBL6260659 0.80 ESR1 (0.59) MAPTPOLBTP53THRBTDP1
SCHEMBL6212239 0.78 POLB (0.50) MAPTPOLBTP53THRBTDP1
SCHEMBL17242043 0.77 MAPT (0.68) MAPTPOLBTP53THRBTDP1
SCHEMBL6211828 0.77 PPARG (0.52) MAPTPOLBTP53THRBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1368324-A1 QUINAZOLINES AS MMP-13 INHIBITORS Warner-Lambert Company LLC (US) 2003-12-10 EP claimed
US-20020193377-A1 Quinazolines as MMP-13 inhibitors ANDRIANJARA CHARLES (FR) 2002-12-19 US claimed
WO-2002064572-A1 QUINAZOLINES AS MMP-13 INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2002-08-22 WO claimed
CN-1537105-A Quinazolines useful as MMP-13 inhibitors ��������ʲ��������ι�˾ 2004-10-13 CN disclosed
US-20020193377-A1 Quinazolines as MMP-13 inhibitors ANDRIANJARA CHARLES (FR) 2002-12-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020193377-A1 Quinazolines as MMP-13 inhibitors MMP13, MMP9, MMP3 MAPT 4823/4885POLB 1104/4885TP53 4351/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.