SCHEMBL7097608

SCHEMBL7097608

Cn1c(=O)n(Cc2cccc(F)c2)c(=O)c2cc(C(=O)O)ncc21

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.47
GRIN1 Q05586 3/20 0.46
GRIN2B Q13224 3/20 0.46
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
HPGD P15428 1/20 0.45
TSHR P16473 1/20 0.45
HTT P42858 1/20 0.45
ATM Q13315 1/20 0.45
MMP13 P45452 1/20 0.44
SLC22A8 Q8TCC7 1/20 0.44
PCSK9 Q8NBP7 1/20 0.44
PARG Q86W56 1/20 0.44
FEN1 P39748 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6255569 0.89 MMP13 (0.53) ALDH1A1HPGDTSHRHTTMMP13
SCHEMBL7018710 0.88 MMP13 (0.46) MAPTALDH1A1LMNAMMP13SLC22A8
SCHEMBL7014083 0.88 MAPK1 (0.55) MAPTALDH1A1LMNAHPGDTSHR
SCHEMBL7022157 0.88 MAPT (0.53) MAPTALDH1A1LMNAHPGDTSHR
SCHEMBL7018972 0.86 GRIN1 (0.44) GRIN1GRIN2BMMP13SLC22A8PARG
SCHEMBL7017009 0.86 MAPT (0.51) MAPTALDH1A1LMNATSHRHTT
SCHEMBL7102299 0.84 GRIN1 (0.44) GRIN1GRIN2BMMP13SLC22A8
SCHEMBL7103058 0.83 MMP13 (0.47) MAPTALDH1A1LMNAHPGDTSHR
SCHEMBL6255189 0.82 MMP13 (0.58) MAPTALDH1A1HTTMMP13SLC22A8
SCHEMBL7097739 0.82 MMP13 (0.46) MAPTALDH1A1LMNAHPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1368324-A1 QUINAZOLINES AS MMP-13 INHIBITORS Warner-Lambert Company LLC (US) 2003-12-10 EP disclosed
US-20020193377-A1 Quinazolines as MMP-13 inhibitors ANDRIANJARA CHARLES (FR) 2002-12-19 US disclosed
WO-2002064572-A1 QUINAZOLINES AS MMP-13 INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2002-08-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020193377-A1 Quinazolines as MMP-13 inhibitors MMP13, MMP9, MMP3 MAPT 4823/4885GRIN1 2546/4885GRIN2B 2437/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.