SCHEMBL7098387

SCHEMBL7098387

CCOc1cc(C2CCCCCN2NC)cnc1Br

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.41
CHRNA4 P43681 1/20 0.41
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
CASP1 P29466 1/20 0.35
CASP7 P55210 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HSD17B10 Q99714 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
POLB P06746 2/20 0.32
OPRK1 P41145 5/20 0.32
APOBEC3G Q9HC16 1/20 0.32
MITF O75030 1/20 0.31
THRB P10828 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7102513 0.99 CHRNB2 (0.42) CHRNB2CHRNA4KDM4EALDH1A1HPGD
SCHEMBL7098316 0.95 CHRNB2 (0.43) CHRNB2CHRNA4KDM4EALDH1A1HPGD
SCHEMBL7101256 0.81 CHRNB2 (0.35) CHRNB2CHRNA4ALDH1A1OPRK1
SCHEMBL7100521 0.81 OPRK1 (0.31) ALDH1A1OPRK1
SCHEMBL7102546 0.79 ALDH1A1 (0.31) CHRNB2CHRNA4KDM4EALDH1A1
SCHEMBL7100526 0.79 CHRNB2 (0.36) CHRNB2CHRNA4ALDH1A1
SCHEMBL7103730 0.78 CHRNB2 (0.41) CHRNB2CHRNA4KDM4EALDH1A1HPGD
SCHEMBL7101803 0.78 CHRNB2 (0.41) CHRNB2CHRNA4KDM4EALDH1A1HPGD
SCHEMBL7098379 0.77 ALDH1A1 (0.44) CHRNB2CHRNA4ALDH1A1OPRK1
SCHEMBL7099495 0.76 CHRNB2 (0.39) CHRNB2CHRNA4KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003500402-A 2003-01-07 JP claimed
EP-1178982-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2002-02-13 EP claimed
WO-2000071534-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2000-11-30 WO claimed
EP-1178982-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2002-02-13 EP disclosed
WO-2000071534-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2000-11-30 WO disclosed