SCHEMBL7098474

SCHEMBL7098474

CC(=COc1ccc(N)cc1)C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.39
PARP10 Q53GL7 1/20 0.39
TDP1 Q9NUW8 6/20 0.39
MAPK1 P28482 1/20 0.39
CYP3A4 P08684 4/20 0.38
ALDH1A1 P00352 4/20 0.38
AKR1C3 P42330 1/20 0.37
TSHR P16473 4/20 0.37
MAOA P21397 2/20 0.36
MAPT P10636 3/20 0.35
TEAD4 Q15561 1/20 0.35
POLB P06746 1/20 0.34
LMNA P02545 2/20 0.34
CYP1A2 P05177 2/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
PDE4D Q08499 1/20 0.34
SMN1; SMN2 Q16637 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2811460 0.83 LMNA (0.48) TDP1CYP3A4ALDH1A1AKR1C3TSHR
SCHEMBL2581335 0.83 AKR1C3 (0.38) PARP10ALDH1A1AKR1C3MAPTRAB9A
SCHEMBL2808566 0.83 CA1 (0.48) PARP10MAPK1ALDH1A1MAPTLMNA
SCHEMBL219559 0.83 AKR1C3 (0.38) PARP10ALDH1A1AKR1C3MAPTRAB9A
SCHEMBL2808572 0.83 CA1 (0.48) PARP10MAPK1ALDH1A1MAPTLMNA
SCHEMBL2811454 0.83 LMNA (0.48) TDP1CYP3A4ALDH1A1AKR1C3TSHR
SCHEMBL156818 0.82 AKR1C3 (0.50) ALDH1A1AKR1C3MAPTCYP2C9
SCHEMBL821031 0.82 AKR1C3 (0.50) ALDH1A1AKR1C3MAPTCYP2C9
SCHEMBL2808898 0.82 CYP2C9 (0.42) MAPK1POLBNPC1RAB9ACYP2C9
SCHEMBL2808895 0.82 CYP2C9 (0.42) MAPK1POLBNPC1RAB9ACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0994911-B1 PROCESS FOR PRODUCING AN ADHERENT POLYMERIC LAYER ON POLYMERIC SUBSTRATES AND ARTICLES PRODUCED THEREBY PPG IND OHIO INC (US) 2003-08-27 EP disclosed
EP-0994911-A1 PROCESS FOR PRODUCING AN ADHERENT POLYMERIC LAYER ON POLYMERIC SUBSTRATES AND ARTICLES PRODUCED THEREBY PPG Industries Ohio, Inc. (US) 2000-04-26 EP disclosed
US-6025026-A POLYMER LAYER ON POLYMER SUBSTRATES WITH REACTIVE SUBSTRATES AND POLYMERIZATION TRANSITIONS OPTICAL, INC. (US) 2000-02-15 US disclosed
WO-1999000448-A1 PROCESS FOR PRODUCING AN ADHERENT POLYMERIC LAYER ON POLYMERIC SUBSTRATES AND ARTICLES PRODUCED THEREBY TRANSITIONS OPTICAL, INC. (US) 1999-01-07 WO disclosed
US-5744243-A ANTIREFLECTIVE SURFACE PPG INDUSTRIES, INC. (US) 1998-04-28 US disclosed
US-5580819-A COATING SUBSTRATE WITH MIXTURE OF PRODUCTS OF ACID-CATALYZED HYDROLYSIS AND CONDENSATION OF SILANE MONOMERS, WATER AND COMPATIBLE FILM FORMING POLYMERS, CURING, THEN TREATING THE COATING WITH AQUEOUS INORGANIC ELECTROLYTE FOR POROSITY PPG INDUSTRIES, INC. (US) 1996-12-03 US disclosed
WO-1996029154-A1 COATING COMPOSITION, PROCESS FOR PRODUCING ANTIREFLECTIVE COATINGS, AND COATED ARTICLES PPG INDUSTRIES, INC. (US) 1996-09-26 WO disclosed
US-5330686-A Crosslinked acrylic ester polymer, benzoxazine compound PPG INDUSTRIES, INC. (US) 1994-07-19 US disclosed
WO-1994004952-A1 TEMPERATURE STABLE AND SUNLIGHT PROTECTED PHOTOCHROMIC ARTICLES PPG INDUSTRIES, INC. (US) 1994-03-03 WO disclosed