SCHEMBL7099030

SCHEMBL7099030

N=C(N)Nc1cccc(C(=O)NNC(=O)CC(CC(=O)O)c2cccc([N+](=O)[O-])c2)c1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 14/20 0.52
ITGAV P06756 14/20 0.52
POLB P06746 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
ITGA2B P08514 3/20 0.47
LMNA P02545 1/20 0.46
MEN1 O00255 1/20 0.46
MAPT P10636 1/20 0.46
BLM P54132 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7262415 0.91 ITGB3 (0.52) ITGB3ITGAVPOLBCYP1A2CYP3A4
SCHEMBL7105696 0.91 ITGB3 (0.51) ITGB3ITGAVPOLBCYP1A2CYP3A4
SCHEMBL7099298 0.88 ITGB3 (0.66) ITGB3ITGAVITGA2B
SCHEMBL7099027 0.84 KDM4E (0.47) ITGB3ITGAVPOLBITGA2BLMNA
SCHEMBL7105309 0.82 ITGB3 (0.68) ITGB3ITGAVITGA2BMEN1KMT2A
SCHEMBL7099697 0.82 ITGB3 (0.68) ITGB3ITGAVITGA2B
SCHEMBL7103664 0.82 ITGB3 (0.68) ITGB3ITGAVITGA2BMEN1KMT2A
SCHEMBL13703191 0.82 ITGB3 (0.57) ITGB3ITGAVITGA2B
SCHEMBL7104742 0.82 ITGB3 (0.68) ITGB3ITGAVITGA2BKMT2A
SCHEMBL7102231 0.82 ITGB3 (0.68) ITGB3ITGAVITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6649613-B1 Integrin inhibitors MERCK PATENT GMBH (DE) 2003-11-18 US disclosed
EP-1194401-B1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2003-09-10 EP disclosed
EP-1194401-A1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GmbH (DE) 2002-04-10 EP disclosed
WO-2001005753-A1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2001-01-25 WO disclosed