SCHEMBL7100276

SCHEMBL7100276

C=CC(O)c1ccc(C#N)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.43
CA2 P00918 3/20 0.43
CA12 O43570 1/20 0.43
CA3 P07451 1/20 0.43
CA6 P23280 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
CYP19A1 P11511 8/20 0.40
MMP3 P08254 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
ALDH1A1 P00352 1/20 0.38
CYP2A6 P11509 1/20 0.38
GSK3B P49841 1/20 0.37
CA1 P00915 2/20 0.36
TSHR P16473 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
CYP2C19 P33261 1/20 0.36
HDAC8 Q9BY41 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12289097 0.79 CA2 (0.43) ENPP2CA2CA12CA3CA6
SCHEMBL6163795 0.77 ENPP2 (0.46) ENPP2ALDH1A1GSK3BTSHRMAPT
SCHEMBL27520915 0.76 CYP19A1 (0.48) ENPP2CA2CA12CA3CA6
SCHEMBL691258 0.75 CA2 (0.52) ENPP2CA2CA12CA3CA6
SCHEMBL3696286 0.75 CA2 (0.52) ENPP2CA2CA12CA3CA6
SCHEMBL26162676 0.75 CA2 (0.52) ENPP2CA2CA12CA3CA6
SCHEMBL2964706 0.75 HRH3 (0.43) ENPP2CA2CA12CA3CA6
SCHEMBL31192685 0.74 MAP2K1 (0.33) ENPP2CA2CA12CA3CA6
SCHEMBL387119 0.73 ESR1 (0.44) CA2CA12CA3CA9CA14
SCHEMBL28387350 0.72 CA12 (0.41) CA2CA12CA3CA6CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113666925-B Method for synthesizing isoindolo [2,1-b ] isoquinoline-5 (7H) -ketone compound 广州大学 2022-05-17 CN disclosed
CN-113666925-A Method for synthesizing isoindolo [2,1-b ] isoquinoline-5 (7H) -ketone compound 广州大学 2021-11-19 CN disclosed
US-20030065176-A1 Factor xa inhibitors with aryl-amidines and derivatives, and prodrugs thereof LG CHEM INVESTMENT LTD. (KR) 2003-04-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030065176-A1 Factor xa inhibitors with aryl-amidines and derivatives, and prodrugs thereof F2, F12, TFPI ENPP2 455/4885CA2 1203/4885CA12 1610/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.