SCHEMBL7101926

SCHEMBL7101926

CNc1cc(C(F)(F)F)cc(C(=O)O)c1C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TAS2R14 Q9NYV8 4/20 0.40
AKR1C3 P42330 2/20 0.37
AKR1C2 P52895 2/20 0.37
RXRA P19793 7/20 0.37
NR1H2 P55055 6/20 0.37
NR1H3 Q13133 4/20 0.37
GPR35 Q9HC97 2/20 0.36
RXRB P28702 1/20 0.36
KDM4E B2RXH2 1/20 0.36
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSD17B10 Q99714 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
LIPC P11150 1/20 0.35
LIPG Q9Y5X9 1/20 0.35
NOTUM Q6P988 1/20 0.35
GRIK1 P39086 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5553664 0.81 KDM4E (0.49) TAS2R14AKR1C3AKR1C2RXRANR1H2
SCHEMBL15920582 0.73 KDM4E (0.54) RXRANR1H2NR1H3RXRBKDM4E
SCHEMBL29756075 0.73 KDM4E (0.54) RXRANR1H2NR1H3RXRBKDM4E
SCHEMBL4417351 0.73 KDM4E (0.54) RXRANR1H2NR1H3KDM4EUSP2
SCHEMBL8570209 0.72 RXRA (0.41) RXRANR1H2NR1H3RXRBKDM4E
SCHEMBL28740934 0.71 CFTR (0.57) RXRANR1H2NR1H3KDM4EALDH1A1
SCHEMBL3886144 0.70 LIPC (0.58) TAS2R14AKR1C3AKR1C2KDM4EUSP2
SCHEMBL22525059 0.70 TAS2R14 (0.58) TAS2R14AKR1C3AKR1C2KDM4EUSP2
SCHEMBL686427 0.69 RXFP1 (0.58) TAS2R14AKR1C3AKR1C2KDM4EUSP2
SCHEMBL1452551 0.69 GRIK1 (0.55) TAS2R14AKR1C3AKR1C2KDM4EUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1343751-A2 CYCLIC DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL-MYERS SQUIBB COMPANY (US) 2003-09-17 EP disclosed
WO-2002060859-A2 CYCLIC DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL-MYERS SQUIBB COMPANY (US) 2002-08-08 WO disclosed