SCHEMBL7102335

SCHEMBL7102335

N=C(N)NCCCCC(=O)NNC(=O)CC(CC(=O)O)c1ccc(Cl)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 12/20 0.61
ITGAV P06756 12/20 0.61
ITGA2B P08514 5/20 0.49
ITGB5 P18084 2/20 0.48
ITGB6 P18564 2/20 0.48
GABBR2 O75899 3/20 0.47
GABBR1 Q9UBS5 3/20 0.47
LMNA P02545 2/20 0.47
CYP2C9 P11712 2/20 0.47
THRB P10828 2/20 0.47
CYP3A4 P08684 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
NFKB1 P19838 1/20 0.47
DRD3 P35462 1/20 0.47
BLM P54132 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47
MEN1 O00255 1/20 0.47
TSHR P16473 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7100423 0.90 ITGB3 (0.61) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL7100379 0.89 ITGB3 (0.60) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL7103319 0.79 ITGB3 (0.46) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL341098 0.77 GABBR2 (0.60) ITGB3ITGAVITGA2BGABBR2GABBR1
Hydrochloric Acid SCHEMBL7076939 0.76 GABBR2 (0.59) ITGB3ITGAVITGA2BGABBR2GABBR1
SCHEMBL7267221 0.74 ITGB3 (0.86) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL7262407 0.74 ITGB3 (0.86) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL12259092 0.73 ITGB3 (0.68) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL7105309 0.72 ITGB3 (0.68) ITGB3ITGAVITGA2BMEN1KMT2A
SCHEMBL391659 0.71 GABBR2 (0.79) GABBR2GABBR1LMNACYP2C9THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6649613-B1 Integrin inhibitors MERCK PATENT GMBH (DE) 2003-11-18 US disclosed
EP-1194401-B1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2003-09-10 EP disclosed