SCHEMBL7100423

SCHEMBL7100423

N=C(N)NCCCCC(=O)NNC(=O)CC(CC(=O)O)c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 15/20 0.61
ITGAV P06756 13/20 0.61
ITGA2B P08514 6/20 0.54
ITGB5 P18084 3/20 0.50
ITGB6 P18564 3/20 0.50
KDM4E B2RXH2 1/20 0.46
RECQL P46063 1/20 0.46
MAPT P10636 1/20 0.46
GABBR2 O75899 1/20 0.43
GABBR1 Q9UBS5 1/20 0.43
APEX1 P27695 1/20 0.43
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7102335 0.90 ITGB3 (0.61) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL7100379 0.85 ITGB3 (0.60) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL12259092 0.83 ITGB3 (0.68) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL7099770 0.77 ITGB3 (0.47) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL8619040 0.75 ITGB3 (0.52) ITGB3ITGAVITGA2BITGB5ITGB6
Hydrochloric Acid SCHEMBL6947022 0.74 GABBR2 (0.56) ITGB3ITGA2BKDM4ERECQLMAPT
SCHEMBL29050822 0.72 MAPT (0.59) ITGB3ITGAVKDM4ERECQLMAPT
SCHEMBL12026728 0.72 ITGB3 (0.54) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL7104922 0.72 ITGB3 (0.89) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL7099298 0.70 ITGB3 (0.66) ITGB3ITGAVITGA2BKDM4ERECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6649613-B1 Integrin inhibitors MERCK PATENT GMBH (DE) 2003-11-18 US claimed
EP-1194401-B1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2003-09-10 EP claimed
US-6649613-B1 Integrin inhibitors MERCK PATENT GMBH (DE) 2003-11-18 US disclosed