SCHEMBL7102474

SCHEMBL7102474

CNCCOc1cncnc1

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.62
CHRNA4 P43681 2/20 0.62
HTR1B P28222 4/20 0.53
HTR1D P28221 2/20 0.53
CDC7 O00311 1/20 0.42
ROCK2 O75116 1/20 0.42
MAP4K4 O95819 1/20 0.42
PIM1 P11309 1/20 0.42
PRKACA P17612 1/20 0.42
CDK2 P24941 1/20 0.42
GSK3B P49841 1/20 0.42
HIPK2 Q9H2X6 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA7 P36544 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7102684 0.79 DRD2 (0.42) CHRNB2CHRNA4
SCHEMBL30756567 0.77 CHRNB2 (1.00) CHRNB2CHRNA4HTR1BHTR1D
SCHEMBL29244418 0.77 CHRNB2 (0.40) CHRNB2CHRNA4HTR1BHTR1DCHRNB4
SCHEMBL7101352 0.77 CHRNB2 (1.00) CHRNB2CHRNA4HTR1BHTR1D
SCHEMBL10158177 0.76 CA12 (0.42) CHRNB2CHRNA4KDM4EALDH1A1CHRNB4
SCHEMBL1935365 0.75 HTR1B (0.64) CHRNB2CHRNA4HTR1BHTR1DKDM4E
SCHEMBL24271048 0.74 CYP2D6 (0.52) KDM4EALDH1A1LMNA
SCHEMBL30625798 0.74 CHRNB2 (0.41) CHRNB2CHRNA4ALDH1A1
SCHEMBL19744084 0.73 MTNR1A (0.45) ALDH1A1LMNA
SCHEMBL7547843 0.72 CHRNB2 (0.39) CHRNB2CHRNA4HTR1BHTR1DALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003500393-A 2003-01-07 JP claimed
EP-1185513-A2 ARYL SUBSTITUTED ALKYLAMINES CAPABLE OF ACTIVATING NICOTINIC CHOLINERGIC RECEPTORS Targacept, Inc. (US) 2002-03-13 EP claimed
WO-2000071520-A2 ARYL SUBSTITUTED ALKYLAMINES CAPABLE OF ACTIVATING NICOTINIC CHOLINERGIC RECEPTORS TARGACEPT, INC. (US) 2000-11-30 WO claimed