SCHEMBL7103221

SCHEMBL7103221

Cc1ccc(C(=O)NNC(=O)c2ccc(C)cc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 1.00
GAA P10253 1/20 1.00
TDP1 Q9NUW8 1/20 0.70
HDAC1 Q13547 1/20 0.70
HDAC6 Q9UBN7 1/20 0.70
HTT P42858 2/20 0.66
RAB9A P51151 5/20 0.64
NPC1 O15118 4/20 0.64
SMN1; SMN2 Q16637 3/20 0.63
KDM4E B2RXH2 1/20 0.63
CCR6 P51684 1/20 0.61
PTGS2 P35354 2/20 0.60
CYP3A4 P08684 1/20 0.59
MAPT P10636 1/20 0.59
CYP2C9 P11712 1/20 0.59
ALOX12 P18054 1/20 0.59
CYP2C19 P33261 1/20 0.59
LMNA P02545 1/20 0.59
CES2 O00748 1/20 0.59
CES1 P23141 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5166735 0.91 ALDH1A1 (0.83) ALDH1A1GAATDP1HTTRAB9A
SCHEMBL13427112 0.91 ALDH1A1 (0.83) ALDH1A1GAATDP1HDAC1HDAC6
SCHEMBL28357030 0.91 ALDH1A1 (0.83) ALDH1A1GAATDP1HDAC1HDAC6
SCHEMBL15964221 0.89 ALDH1A1 (0.79) ALDH1A1GAATDP1HDAC1HDAC6
SCHEMBL19663861 0.88 ALDH1A1 (0.78) ALDH1A1GAATDP1HDAC1HDAC6
SCHEMBL13381492 0.87 ALDH1A1 (0.76) ALDH1A1GAATDP1HDAC1HDAC6
SCHEMBL2896135 0.87 ALDH1A1 (0.76) ALDH1A1GAATDP1HDAC1HDAC6
SCHEMBL8726176 0.85 ALDH1A1 (0.73) ALDH1A1GAATDP1HDAC1HDAC6
SCHEMBL31375604 0.85 GAA (0.73) ALDH1A1GAATDP1HDAC1HDAC6
SCHEMBL14527271 0.85 CTDSP1 (0.78) ALDH1A1GAAHDAC1HTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1135363-B1 PROCESS FOR THE PREPARATION OF SYMMETRICAL DIACYLHYDRAZINES GREAT LAKES CHEMICAL EUROP (CH) 2003-09-24 EP claimed
US-6444848-B1 REACTING HYDRAZINE WITH ACID CHLORIDE GREAT LAKES CHEMICAL (EUROPE) GMBH (DE) 2002-09-03 US claimed
EP-1135363-A1 PROCESS FOR THE PREPARATION OF SYMMETRICAL DIACYLHYDRAZINES Great Lakes Chemical (Europe) GmbH (CH) 2001-09-26 EP claimed
WO-2000034227-A1 PROCESS FOR THE PREPARATION OF SYMMETRICAL DIACYLHYDRAZINES GREAT LAKES CHEMICAL (EUROPE) GMBH (CH) 2000-06-15 WO claimed
US-8908132-B2 Blue phase mode liquid crystal display device and method of manufacturing the same LG DISPLAY CO., LTD. (KR) 2014-12-09 US disclosed
US-8848156-B2 Liquid crystal display device LG DISPLAY CO., LTD. (KR) 2014-09-30 US disclosed
US-8045117-B2 Display element and display device SHARP KABUSHIKI KAISHA (JP) 2011-10-25 US disclosed
US-20110141421-A1 LIQUID CRYSTAL DISPLAY DEVICE LG DISPLAY CO., LTD. (KR) 2011-06-16 US disclosed
US-20110141415-A1 BLUE PHASE MODE LIQUID CRYSTAL DISPLAY DEVICE AND METHOD OF MANUFACTURING THE SAME LG DISPLAY CO., LTD. (KR) 2011-06-16 US disclosed
US-20100014040-A1 Display element and display device SHARP KABUSHIKI KAISHA (JP) 2010-01-21 US disclosed
EP-1135363-B1 PROCESS FOR THE PREPARATION OF SYMMETRICAL DIACYLHYDRAZINES GREAT LAKES CHEMICAL EUROP (CH) 2003-09-24 EP disclosed
US-6444848-B1 REACTING HYDRAZINE WITH ACID CHLORIDE GREAT LAKES CHEMICAL (EUROPE) GMBH (DE) 2002-09-03 US disclosed
EP-1135363-A1 PROCESS FOR THE PREPARATION OF SYMMETRICAL DIACYLHYDRAZINES Great Lakes Chemical (Europe) GmbH (CH) 2001-09-26 EP disclosed
WO-2000034227-A1 PROCESS FOR THE PREPARATION OF SYMMETRICAL DIACYLHYDRAZINES GREAT LAKES CHEMICAL (EUROPE) GMBH (CH) 2000-06-15 WO disclosed
US-4052362-A N-CINNAMOYL-N'-ACYLHYDRAZINES UBE INDUSTRIES, LTD. (JA) 1977-10-04 US disclosed
US-4043976-A N,N'-DIBENZOYLHYDRAZINE DERIVATIVE UBE INDUSTRIES, LTD. (JA) 1977-08-23 US disclosed