SCHEMBL7105261

SCHEMBL7105261

CC(C)(C)OC(=O)c1cccnc1C1=CCNCC1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
POLB P06746 1/20 0.37
SIGMAR1 Q99720 1/20 0.36
HTR2C P28335 1/20 0.35
QDPR P09417 2/20 0.35
HTR6 P50406 2/20 0.35
GRM5 P41594 1/20 0.35
GRM1 Q13255 1/20 0.35
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
HTR2A P28223 1/20 0.35
HTR7 P34969 1/20 0.35
FTO Q9C0B1 1/20 0.34
KDM4E B2RXH2 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
BRPF1 P55201 1/20 0.34
CDK9 P50750 4/20 0.33
CCNT1 O60563 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30469414 1.00 ADRA1A (0.39) ADRA1AADRA1BPOLBSIGMAR1HTR2C
SCHEMBL4294398 0.72 SCN9A (0.39) SIGMAR1HTR2CQDPRCDK9
SCHEMBL4004663 0.72 SIGMAR1 (0.47) SIGMAR1HTR2CQDPRHTR6GRM5
SCHEMBL30617923 0.71 TDP1 (0.41) ADRA1AADRA1BPOLBKDM4ETDP1
SCHEMBL31652073 0.71 CCNT1 (0.50) SIGMAR1HTR2CQDPRCDK9CCNT1
Trifluoroacetic Acid SCHEMBL3854727 0.70 TRPV1 (0.40) SIGMAR1HTR2C
SCHEMBL2428360 0.70 GRM5 (0.57) POLBGRM5GRM1
SCHEMBL13228917 0.69 CDK9 (0.47) SIGMAR1HTR2CQDPRGRM5KDM4E
SCHEMBL4004617 0.69 SIGMAR1 (0.49) SIGMAR1HTR2CQDPRHTR6GRM5
SCHEMBL7454398 0.69 SIGMAR1 (0.47) SIGMAR1HTR2CQDPRGRM5CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003101994-A1 FUSED BICYCLIC AROMATIC COMPOUNDS THAT ARE USEFUL IN TREATING SEXUAL DYSFUNCTION ABBOTT LABORATORIES (US) 2003-12-11 WO disclosed