SCHEMBL7105342

SCHEMBL7105342

CN1CCN(c2c(-c3ccc(Cl)cc3Cl)ncc(CCN3CCCC3)c2N)C(=O)C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.43
GSK3A P49840 1/20 0.43
EPHX2 P34913 1/20 0.37
CNR1 P21554 5/20 0.36
OPRM1 P35372 1/20 0.35
OPRK1 P41145 1/20 0.35
HTR2C P28335 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C19 P33261 1/20 0.35
MCHR1 Q99705 1/20 0.35
CNR2 P34972 1/20 0.34
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
DPP4 P27487 1/20 0.33
DPP8 Q6V1X1 1/20 0.33
DPP9 Q86TI2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13211502 0.64 GSK3B (0.47) GSK3BGSK3APOLBCYP3A4SLC6A2
SCHEMBL2911529 0.63 MAPT (0.45) GSK3BGSK3ATDP1ALDH1A1
SCHEMBL7105334 0.61 SLC6A2 (0.33) GSK3BGSK3AHTR2CTDP1KDM4E
SCHEMBL3598377 0.60 DPP4 (0.43) CNR1TDP1CYP3A4CYP2C19MCHR1
SCHEMBL3598863 0.60 HTT (0.43) CNR1TDP1CYP3A4CYP2C19MCHR1
SCHEMBL27559805 0.59 POLB (0.50) CNR1KDM4EPOLB
SCHEMBL157609 0.59 SLC6A2 (0.56) ALDH1A1POLBSLC6A2SLC6A4
SCHEMBL21424922 0.58 DRD2 (0.57) ALDH1A1SLC6A2SLC6A4
SCHEMBL20200690 0.57 HRH3 (0.42)
SCHEMBL27538115 0.57 CYP2A13 (0.55) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317433-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2003-06-11 EP disclosed
WO-2002020495-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2002-03-14 WO disclosed