SCHEMBL7105936

SCHEMBL7105936

CC(C)(C)OC(=O)N[C@H](C(=O)O)[C@H](OC(=O)c1ccccc1)C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.55
TP53 P04637 1/20 0.55
PPARA Q07869 6/20 0.48
PPARG P37231 5/20 0.48
ATM Q13315 1/20 0.47
RECQL P46063 1/20 0.46
PPARD Q03181 2/20 0.46
CYP2D6 P10635 1/20 0.45
APP P05067 2/20 0.43
ALDH1A1 P00352 1/20 0.42
HSD17B10 Q99714 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
CTSK P43235 2/20 0.41
CTSS P25774 2/20 0.41
ACE P12821 1/20 0.41
JAK3 P52333 1/20 0.40
BTK Q06187 1/20 0.40
ADRB2 P07550 1/20 0.40
ADRB1 P08588 1/20 0.40
ADRB3 P13945 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7105931 1.00 TSHR (0.55) TSHRTP53PPARAPPARGATM
SCHEMBL7097578 0.87 GABRB1 (0.54) TSHRTP53PPARAPPARGATM
SCHEMBL7097577 0.87 GABRB1 (0.54) TSHRTP53PPARAPPARGATM
SCHEMBL9544071 0.86 PPARA (0.46) TSHRTP53PPARAPPARGATM
SCHEMBL9544068 0.86 PPARA (0.46) TSHRTP53PPARAPPARGATM
SCHEMBL30496988 0.80 ATM (0.48) TSHRTP53PPARAPPARGATM
SCHEMBL30158979 0.79 TSHR (0.69) TSHRTP53RECQLCYP2D6ALDH1A1
SCHEMBL7105585 0.78 CTSK (0.43) PPARAPPARGATMCYP2D6CTSK
SCHEMBL7105576 0.78 CTSK (0.43) PPARAPPARGATMCYP2D6CTSK
SCHEMBL7099862 0.77 PPARA (0.58) PPARAPPARGATMPPARDCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0990640-B1 Beta-Hydroxyaspartic acid derivatives SUNTORY LTD (JP) 2003-01-22 EP disclosed
EP-0844234-B1 Beta-hydroxyaspartic acid derivatives SUNTORY LTD (JP) 2002-03-06 EP disclosed
US-6147113-A ADMINISTERING TO TREAT NERVOUS SYSTEM AND BRAIN DISORDERS; GLUTAMATE UPTAKE INHIBITORS SUNTORY LIMITED (JP) 2000-11-14 US disclosed
EP-0990640-A2 Beta-Hydroxyaspartic acid derivatives SUNTORY LIMITED (JP) 2000-04-05 EP disclosed
EP-0948962-A2 Beta-hydroxyaspartic acid derivatives SUNTORY LIMITED (JP) 1999-10-13 EP disclosed
EP-0844234-A2 Beta-hydroxyaspartic acid derivatives SUNTORY LIMITED (JP) 1998-05-27 EP disclosed