SCHEMBL7106614

SCHEMBL7106614

COc1cc(CN2C(=O)N([C@@H](CC(C)C)C(=O)O)C(=O)C23CCCCC3)ccc1NC(=O)Nc1ccccc1C

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 13/20 0.44
ITGB1 P05556 12/20 0.44
CHEK1 O14757 2/20 0.38
LPAR1 Q92633 1/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
ATM Q13315 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7106166 0.88 ITGB1 (0.45) ITGA4ITGB1
SCHEMBL4671791 0.88 ITGA4 (0.47) ITGA4ITGB1CHEK1LPAR1MEN1
SCHEMBL4671784 0.88 ITGA4 (0.47) ITGA4ITGB1CHEK1LPAR1MEN1
SCHEMBL7382803 0.88 ITGB1 (0.45) ITGA4ITGB1ATM
SCHEMBL1817892 0.88 ITGB1 (0.45) ITGA4ITGB1ATM
SCHEMBL1825903 0.88 ITGB1 (0.45) ITGA4ITGB1ATM
SCHEMBL6165813 0.85 ITGA4 (0.45) ITGA4ITGB1CHEK1LPAR1MEN1
Tromethamine SCHEMBL1820966 0.83 ITGB1 (0.41) ITGA4ITGB1
SCHEMBL7101082 0.81 ITGB1 (0.49) ITGA4ITGB1
SCHEMBL7102059 0.81 ITGB1 (0.49) ITGA4ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183241-B1 SPIROIMIDAZOLIDINE DERIVATIVES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL PREPARATIONS COMPRISING THEM AVENTIS PHARMA GMBH (DE) 2003-09-17 EP disclosed
US-6399643-B1 ANTIINFLAMMATORY AGENTS; ANTIARTHRITIC AGENTS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2002-06-04 US disclosed
EP-1183241-A1 SPIROIMIDAZOLIDINE DERIVATIVES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL PREPARATIONS COMPRISING THEM Aventis Pharma Deutschland GmbH (DE) 2002-03-06 EP disclosed
WO-2000069831-A1 SPIROIMIDAZOLIDINE DERIVATIVES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL PREPARATIONS COMPRISING THEM AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-11-23 WO disclosed