SCHEMBL7107701

SCHEMBL7107701

COc1cccc(-c2cc3ccccc3s2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 1/20 0.56
HSD17B2 P37059 1/20 0.56
SMN1; SMN2 Q16637 3/20 0.56
MAPT P10636 2/20 0.56
NFKB1 P19838 2/20 0.56
RAB9A P51151 2/20 0.56
NFKB2 Q00653 2/20 0.56
RELA Q04206 2/20 0.56
TDP1 Q9NUW8 2/20 0.56
APP P05067 2/20 0.54
ALDH1A1 P00352 2/20 0.52
HPGD P15428 2/20 0.52
NPC1 O15118 1/20 0.52
TP53 P04637 1/20 0.52
ALOX15 P16050 1/20 0.52
TSHR P16473 1/20 0.52
MAPK1 P28482 1/20 0.52
HSD17B10 Q99714 1/20 0.52
IKBKB O14920 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7107469 0.87 ESR1 (0.51) SMN1; SMN2MAPTNFKB1RAB9ANFKB2
SCHEMBL6173418 0.87 RAB9A (0.68) HSD17B1HSD17B2SMN1; SMN2MAPTNFKB1
SCHEMBL8266537 0.86 TNFRSF1A (0.56) HSD17B1HSD17B2SMN1; SMN2MAPTNFKB1
SCHEMBL5681616 0.83 ESR1 (0.50) HSD17B1HSD17B2SMN1; SMN2MAPTNFKB1
SCHEMBL27631114 0.82 HSD17B1 (0.77) HSD17B1HSD17B2APPERN1CA1
SCHEMBL9151832 0.82 BACE1 (0.56) SMN1; SMN2MAPTNFKB1RAB9ANFKB2
SCHEMBL6832572 0.82 ESR1 (0.58) SMN1; SMN2MAPTNFKB1RAB9ANFKB2
SCHEMBL163523 0.80 APP (0.71) HSD17B1HSD17B2APPERN1CA1
SCHEMBL29766071 0.80 APP (0.71) HSD17B1HSD17B2APPERN1CA1
Bromide SCHEMBL31564934 0.79 APP (0.69) HSD17B1HSD17B2APPERN1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0827959-B1 Benzo[B]thiophene compounds, intermediates, processes, compositions, and methods LILLY CO ELI (US) 2003-12-03 EP disclosed
US-5977382-A Benzo[b]thiophene compounds, intermediates, processes, compositions, and methods ELI LILLY AND COMPANY (US) 1999-11-02 US disclosed
US-5977098-A Benzo[B]thiophene compounds, intermediates, processes, compositions, and methods ELI LILLY AND COMPANY (US) 1999-11-02 US disclosed
US-5952513-A TREATING POSTMENOPAUSAL SYNDROME SUCH AS OSTEOPOROSIS ELI LILLY AND COMPANY (US) 1999-09-14 US disclosed
US-5843965-A Benzo B! thiophene compounds, intermediates, processes, compositions, and methods ELI LILLY AND COMPANY (US) 1998-12-01 US disclosed
EP-0827959-A2 Benzo[B]thiophene compounds, intermediates, processes, compositions, and methods ELI LILLY AND COMPANY (US) 1998-03-11 EP disclosed