SCHEMBL7108274

SCHEMBL7108274

Cc1cc(Oc2cccc(C(F)(F)F)c2)nc(C(=O)O)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.61
KDM4E B2RXH2 3/20 0.49
RAB9A P51151 1/20 0.49
GAA P10253 2/20 0.47
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
RECQL P46063 1/20 0.46
LRRK2 Q5S007 1/20 0.46
ALDH1A1 P00352 3/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
POLB P06746 1/20 0.45
FFAR4 Q5NUL3 1/20 0.44
MAPK1 P28482 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
P2RY1 P47900 1/20 0.43
NPSR1 Q6W5P4 2/20 0.43
LMNA P02545 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8507324 0.88 MAPT (0.56) MAPTKDM4ERAB9AGAACYP1A2
SCHEMBL8058768 0.88 MAPT (0.76) MAPTKDM4ERAB9AGAACYP1A2
SCHEMBL7049881 0.86 MAPT (0.63) MAPTKDM4ERAB9AGAACYP1A2
SCHEMBL8059054 0.86 MAPT (0.60) MAPTKDM4ERAB9AGAACYP1A2
SCHEMBL7113284 0.85 MAPT (0.62) MAPTKDM4ERAB9AGAACYP1A2
SCHEMBL7108376 0.85 MAPT (0.58) MAPTKDM4EGAALRRK2ALDH1A1
SCHEMBL7107323 0.84 MAPT (0.58) MAPTKDM4ERAB9AGAACYP1A2
SCHEMBL7110920 0.84 MAPT (0.58) MAPTKDM4ERAB9AGAACYP1A2
SCHEMBL7110619 0.84 MAPT (0.74) MAPTKDM4ERAB9AGAACYP1A2
SCHEMBL8074437 0.82 MAPT (0.58) MAPTKDM4ERAB9AGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0949248-B1 6-(NONSUBSTITUTED OR SUBSTITUTED) PHENOXYPICOLINIC ACIDS, PROCESS OF PREPARING THE SAME, AND AGRICULTURAL/HORTICULTURAL GERMICIDES CONTAINING THE SAME KUREHA CHEMICAL IND CO LTD (JP) 2003-10-08 EP disclosed
US-6200933-B1 LOW TOXICITY TO HUMANS AND CATTLE KUREHA KAGAKU KABUSHIKI KAISHA (JP) 2001-03-13 US disclosed
US-6159901-A 6-phenoxy picolinic acid alkylidene hydrazide derivative, process for producing the same and herbicide using the same KUREHA KAGAKU KOGYO KABUSHIKI KAISHA (JP) 2000-12-12 US disclosed
EP-1020444-A1 6-PHENOXYPICOLINIC ACID, ALKYLIDENEHYDRAZIDE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, AND HERBICIDE KUREHA KAGAKU KOGYO KABUSHIKI KAISHA (JP) 2000-07-19 EP disclosed
EP-0949248-A1 6-(NONSUBSTITUTED OR SUBSTITUTED) PHENOXYPICOLINIC ACIDS, PROCESS OF PREPARING THE SAME, AND AGRICULTURAL/HORTICULTURAL GERMICIDES CONTAINING THE SAME KUREHA KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1999-10-13 EP disclosed