SCHEMBL7108376

SCHEMBL7108376

O=C(O)c1cc(Cl)cc(Oc2cccc(C(F)(F)F)c2)n1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.58
PPARG P37231 4/20 0.48
NTRK1 P04629 1/20 0.47
GAA P10253 1/20 0.47
P2RY1 P47900 3/20 0.46
ALDH1A1 P00352 1/20 0.45
POLB P06746 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
KDM4E B2RXH2 1/20 0.44
MRGPRX4 Q96LA9 2/20 0.43
LOXL2 Q9Y4K0 1/20 0.43
LRRK2 Q5S007 1/20 0.43
STK39 Q9UEW8 1/20 0.43
PTGER4 P35408 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8773192 0.88 MAPT (0.52) MAPTPPARGNTRK1GAAP2RY1
SCHEMBL7110627 0.87 MAPT (0.74) MAPTPPARGNTRK1GAAP2RY1
SCHEMBL7108274 0.85 MAPT (0.61) MAPTPPARGNTRK1GAAP2RY1
SCHEMBL7110619 0.84 MAPT (0.74) MAPTPPARGNTRK1GAAALDH1A1
SCHEMBL7049881 0.84 MAPT (0.63) MAPTPPARGNTRK1GAAP2RY1
SCHEMBL7113284 0.83 MAPT (0.62) MAPTNTRK1GAAP2RY1ALDH1A1
SCHEMBL7105791 0.82 MAPT (0.55) MAPTPPARGGAAALDH1A1POLB
SCHEMBL7107323 0.82 MAPT (0.58) MAPTPPARGNTRK1GAAP2RY1
SCHEMBL7110920 0.82 MAPT (0.58) MAPTPPARGNTRK1GAAALDH1A1
SCHEMBL8074437 0.80 MAPT (0.58) MAPTPPARGNTRK1GAAP2RY1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0949248-B1 6-(NONSUBSTITUTED OR SUBSTITUTED) PHENOXYPICOLINIC ACIDS, PROCESS OF PREPARING THE SAME, AND AGRICULTURAL/HORTICULTURAL GERMICIDES CONTAINING THE SAME KUREHA CHEMICAL IND CO LTD (JP) 2003-10-08 EP disclosed
US-6200933-B1 LOW TOXICITY TO HUMANS AND CATTLE KUREHA KAGAKU KABUSHIKI KAISHA (JP) 2001-03-13 US disclosed
US-6159901-A 6-phenoxy picolinic acid alkylidene hydrazide derivative, process for producing the same and herbicide using the same KUREHA KAGAKU KOGYO KABUSHIKI KAISHA (JP) 2000-12-12 US disclosed
EP-1020444-A1 6-PHENOXYPICOLINIC ACID, ALKYLIDENEHYDRAZIDE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, AND HERBICIDE KUREHA KAGAKU KOGYO KABUSHIKI KAISHA (JP) 2000-07-19 EP disclosed
EP-0949248-A1 6-(NONSUBSTITUTED OR SUBSTITUTED) PHENOXYPICOLINIC ACIDS, PROCESS OF PREPARING THE SAME, AND AGRICULTURAL/HORTICULTURAL GERMICIDES CONTAINING THE SAME KUREHA KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1999-10-13 EP disclosed