SCHEMBL7108522

SCHEMBL7108522

CN(CCO)C(=O)c1cnc(C(=O)N(C)CCO)cn1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMO Q99835 2/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
POLB P06746 2/20 0.38
HDAC4 P56524 1/20 0.38
CYP11B2 P19099 1/20 0.36
HTR2C P28335 1/20 0.36
CNR1 P21554 1/20 0.35
LRRK2 Q5S007 1/20 0.34
PDK2 Q15119 2/20 0.34
OPRM1 P35372 1/20 0.34
OPRL1 P41146 1/20 0.34
MAPT P10636 2/20 0.33
PDCD1 Q15116 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
TLR9 Q9NR96 1/20 0.32
TLR8 Q9NR97 1/20 0.32
TLR7 Q9NYK1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18130956 0.90 SIRT6 (0.47) SMOMEN1KMT2APOLBHDAC4
SCHEMBL7655050 0.83 HDAC4 (0.44) HDAC4CYP11B2PDK2TLR9TLR8
SCHEMBL24341942 0.83 TDP1 (0.42) SMOHDAC4HTR2CCNR1MAPT
SCHEMBL20327068 0.81 MTOR (0.39) SMOHDAC4HTR2CLRRK2PDK2
SCHEMBL7107359 0.81 HDAC4 (0.39) SMOKMT2APOLBHDAC4HTR2C
SCHEMBL18348214 0.80 MAPT (0.36) SMOMEN1KMT2AHDAC4HTR2C
SCHEMBL7105124 0.79 L3MBTL1 (0.41) POLBCNR1MAPT
SCHEMBL25094798 0.79 ESRRG (0.41) MEN1KMT2AHDAC4
SCHEMBL24800710 0.79 HDAC4 (0.34) SMOMEN1KMT2AHDAC4CYP11B2
SCHEMBL7652649 0.77 HTR2C (0.46) MEN1KMT2AHDAC4HTR2CCNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001944-B1 PYRAZINE DERIVATIVES, PREPARATION AND MEDICINES CONTAINING THEM AVENTIS PHARMA SA (FR) 2003-10-01 EP claimed