SCHEMBL7112165

SCHEMBL7112165

Cc1ccc(-c2cc(C(F)F)nn2NS(=O)(=O)c2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.51
PTGS1 P23219 4/20 0.51
MAPT P10636 1/20 0.40
NPY5R Q15761 1/20 0.40
ALDH1A1 P00352 2/20 0.39
MCL1 Q07820 1/20 0.39
CYP2C9 P11712 1/20 0.38
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzenesulfonamide SCHEMBL7927040 0.94 PTGS2 (0.60) PTGS2PTGS1ALDH1A1CYP2C9LMNA
SCHEMBL8688860 0.91 PTGS2 (0.52) PTGS2PTGS1
SCHEMBL8635921 0.89 PTGS2 (0.46) PTGS2PTGS1
SCHEMBL8688703 0.88 PTGS2 (0.41) PTGS2PTGS1ALDH1A1
SCHEMBL8618309 0.88 PTGS2 (0.51) PTGS2PTGS1
Benzene SCHEMBL7058431 0.88 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL8688398 0.87 PTGS1 (0.53) PTGS2PTGS1MAPTNPY5RALDH1A1
SCHEMBL8636817 0.87 PTGS2 (0.42) PTGS2PTGS1ALDH1A1
SCHEMBL8639178 0.86 PTGS2 (0.43) PTGS2PTGS1NPY5RALDH1A1CYP2C9
SCHEMBL8689218 0.85 PTGS2 (0.41) PTGS2PTGS1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1299122-A2 COMBINATION OF A COX-2 INHIBITOR AND A VASOMODULATOR FOR TREATING PAIN AND HEADACHE PAIN Pharmacia Corporation (US) 2003-04-09 EP claimed
WO-2002005799-A2 COMBINATION OF A COX-2 INHIBITOR AND A VASOMODULATOR FOR TREATING PAIN AND HEADACHE PAIN PHARMACIA CORPORATION (US) 2002-01-24 WO claimed
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US claimed
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed