SCHEMBL8636817

SCHEMBL8636817

CSc1ccc(-c2cc(C(F)F)nn2NS(=O)(=O)c2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.42
PTGS1 P23219 5/20 0.42
ALDH1A1 P00352 3/20 0.40
MMP2 P08253 2/20 0.39
MMP1 P03956 1/20 0.39
MMP3 P08254 1/20 0.39
MMP13 P45452 1/20 0.39
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
MMP9 P14780 1/20 0.37
ESR1 P03372 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8688860 0.88 PTGS2 (0.52) PTGS2PTGS1MMP2MMP1MMP13
SCHEMBL7112165 0.87 PTGS2 (0.51) PTGS2PTGS1ALDH1A1
SCHEMBL8635921 0.86 PTGS2 (0.46) PTGS2PTGS1
Benzene SCHEMBL7058431 0.85 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL8618309 0.85 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL8688398 0.84 PTGS1 (0.53) PTGS2PTGS1ALDH1A1MMP2MMP1
SCHEMBL8420779 0.84 ALDH1A1 (0.41) PTGS2PTGS1ALDH1A1MMP2MMP1
SCHEMBL8639178 0.83 PTGS2 (0.43) PTGS2PTGS1ALDH1A1MMP2MMP1
SCHEMBL8688703 0.83 PTGS2 (0.41) PTGS2PTGS1ALDH1A1
SCHEMBL8641068 0.83 PTGS2 (0.53) PTGS2PTGS1ALDH1A1GAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US claimed
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed
US-5753688-A ANTIINFLAMMATORY TALLEY JOHN J (US) 1998-05-19 US disclosed
US-5510496-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed