SCHEMBL8639178

SCHEMBL8639178

O=S(=O)(Nn1nc(C(F)F)cc1-c1ccc(C(F)(F)F)cc1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.43
PTGS1 P23219 5/20 0.43
HSD11B1 P28845 1/20 0.42
NPY5R Q15761 1/20 0.42
ACLY P53396 1/20 0.39
S1PR1 P21453 1/20 0.39
PTGES2 Q9H7Z7 2/20 0.39
MMP1 P03956 2/20 0.39
MMP9 P14780 2/20 0.39
MMP13 P45452 2/20 0.39
MMP8 P22894 1/20 0.39
MMP12 P39900 1/20 0.39
MMP14 P50281 1/20 0.39
CYP2C9 P11712 1/20 0.38
ALDH1A1 P00352 2/20 0.38
LMNA P02545 1/20 0.38
PDPK1 O15530 1/20 0.38
MEN1 O00255 1/20 0.37
POLB P06746 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8688860 0.89 PTGS2 (0.52) PTGS2PTGS1MMP1MMP9MMP13
Benzene SCHEMBL7058431 0.86 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL7112165 0.86 PTGS2 (0.51) PTGS2PTGS1NPY5RCYP2C9ALDH1A1
SCHEMBL8618309 0.86 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL8641577 0.86 PTGS2 (0.49) PTGS2PTGS1HSD11B1NPY5RACLY
SCHEMBL8635921 0.85 PTGS2 (0.46) PTGS2PTGS1
SCHEMBL8423929 0.85 NPY5R (0.51) PTGS2PTGS1HSD11B1NPY5RACLY
SCHEMBL8693645 0.83 PTGS2 (0.53) PTGS2PTGS1HSD11B1ACLYPTGES2
SCHEMBL8636817 0.83 PTGS2 (0.42) PTGS2PTGS1MMP1MMP9MMP13
SCHEMBL8688398 0.83 PTGS1 (0.53) PTGS2PTGS1NPY5RMMP1MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed
US-5753688-A ANTIINFLAMMATORY TALLEY JOHN J (US) 1998-05-19 US disclosed
US-5510496-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed